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Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50037026
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113815(4-(2-Naphthalen-1-yl-ethyl)-5-piperidin-4-yl-isoxa...)
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50000687(2-(3-Carboxy-propyl)-6-(4-methoxy-phenyl)-2H-pyrid...)
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113812(4-Benzhydryl-5-piperidin-4-yl-isoxazol-3-ol; hydro...)
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113824(4-Phenethyl-5-piperidin-4-yl-isoxazol-3-ol; hydrob...)
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113817(4-(2-Naphthalen-2-yl-ethyl)-5-piperidin-4-yl-isoxa...)
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113804(4-Anthracen-9-ylmethyl-5-piperidin-4-yl-isoxazol-3...)
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113813(4-Biphenyl-4-ylmethyl-5-piperidin-4-yl-isoxazol-3-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50095533(4-(naphthalen-2-ylmethyl)-5-(piperidin-4-yl)isoxaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113810(4-Naphthalen-1-ylmethyl-5-piperidin-4-yl-isoxazol-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113806(4-(3,3-Diphenyl-propyl)-5-piperidin-4-yl-isoxazol-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113808(4-Benzyl-5-piperidin-4-yl-isoxazol-3-ol; hydrobrom...)
Affinity DataIC50: >1.00E+5nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113821(4-Hexyl-5-piperidin-4-yl-isoxazol-3-ol; hydrobromi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113814(4-Cyclohexylmethyl-5-piperidin-4-yl-isoxazol-3-ol;...)
Affinity DataIC50: >1.00E+5nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113816(4-Octyl-5-piperidin-4-yl-isoxazol-3-ol; hydrobromi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113822(5-(4-Methyl-piperidin-4-yl)-isoxazol-3-ol; hydrobr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113819(4-(4,4-Diphenyl-butyl)-5-piperidin-4-yl-isoxazol-3...)
Affinity DataIC50: >1.00E+5nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113823(4-Butyl-5-piperidin-4-yl-isoxazol-3-ol; hydrobromi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113811(4-(2,2-Diphenyl-ethyl)-5-piperidin-4-yl-isoxazol-3...)
Affinity DataIC50: >1.00E+5nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113818(5-Piperidin-4-yl-4-propyl-isoxazol-3-ol; hydrobrom...)
Affinity DataIC50: >1.00E+5nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113805(4-(3-Phenyl-propyl)-5-piperidin-4-yl-isoxazol-3-ol...)
Affinity DataIC50: >1.00E+5nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113809(4-Ethyl-5-piperidin-4-yl-isoxazol-3-ol; hydrobromi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50113803(4-Methyl-5-piperidin-4-yl-isoxazol-3-ol; hydrobrom...)
Affinity DataIC50: >1.00E+5nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
The Royal Danish School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50032954(5-(piperidin-4-yl)isoxazol-3-ol | 5-Piperidin-4-yl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Affinity for GABA-B receptor by inhibiting GABA uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed