Compile Data Set for Download or QSAR
maximum 50k data
Found 14 of ec50 data for polymerid = 49000854
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032671(6-[1-(3,5,5,8,8-PENTAMETHYL-5,6,7,8-TETRAHYDRONAPH...)
Affinity DataEC50:  11nMAssay Description:In vitro transcriptional activation in CV-1 cells expressing RXR-alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50445060(CHEMBL3098773)
Affinity DataEC50:  19nMAssay Description:Agonist activity at RXR-alpha in rat R3KE cells infected with oncogene KLF4-ER assessed as inhibition of KLF4-mediated oncogenic transformationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at RXRalpha in rat RK3E cells assessed as transcriptional activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataEC50:  110nMAssay Description:Agonist activity at RXR-alpha in rat R3KE cells infected with oncogene KLF4-ER assessed as inhibition of KLF4-mediated oncogenic transformationMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017994(CHEMBL3289658)
Affinity DataEC50:  110nMAssay Description:Agonist activity at RXR-alpha in rat R3KE cells infected with oncogene KLF4-ER assessed as inhibition of KLF4-mediated oncogenic transformationMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50445061(CHEMBL3098772)
Affinity DataEC50:  110nMAssay Description:Agonist activity at RXRalpha in rat RK3E cells assessed as transcriptional activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at RXRalpha in rat RK3E cells assessed as transcriptional activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50445059(CHEMBL3098858)
Affinity DataEC50:  120nMAssay Description:Agonist activity at RXRalpha in rat RK3E cells assessed as transcriptional activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50445060(CHEMBL3098773)
Affinity DataEC50:  120nMAssay Description:Agonist activity at RXRalpha in rat RK3E cells assessed as transcriptional activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50445062(CHEMBL3098771)
Affinity DataEC50:  400nMAssay Description:Agonist activity at RXR-alpha in rat R3KE cells infected with oncogene KLF4-ER assessed as inhibition of KLF4-mediated oncogenic transformationMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50018004(CHEMBL3289657)
Affinity DataEC50:  440nMAssay Description:Agonist activity at RXR-alpha in rat R3KE cells infected with oncogene KLF4-ER assessed as inhibition of KLF4-mediated oncogenic transformationMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50445062(CHEMBL3098771)
Affinity DataEC50:  820nMAssay Description:Agonist activity at RXRalpha in rat RK3E cells assessed as transcriptional activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50018005(CHEMBL3289660)
Affinity DataEC50:  880nMAssay Description:Agonist activity at RXR-alpha in rat R3KE cells infected with oncogene KLF4-ER assessed as inhibition of KLF4-mediated oncogenic transformationMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50018001(CHEMBL3289659)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at RXR-alpha in rat R3KE cells infected with oncogene KLF4-ER assessed as inhibition of KLF4-mediated oncogenic transformationMore data for this Ligand-Target Pair