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Found 1908 Enz. Inhib. hit(s) with Target = 'Neuropeptide Y receptor type 5'
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM141347(US8916594, I-024)
Affinity DataIC50:  0.130nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50390219(CHEMBL2070148)
Affinity DataIC50:  0.160nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50390216(CHEMBL2070151)
Affinity DataIC50:  0.160nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM141350(US8916594, I-034)
Affinity DataIC50:  0.180nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50390213(CHEMBL2069316)
Affinity DataIC50:  0.200nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50258001(CHEMBL492370 | N-(3,4-dichlorophenyl)-1-(methylsul...)
Affinity DataIC50:  0.200nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50093652(2-Methyl-6-pentyl-4-piperidin-1-yl-5H-pyrrolo[3,2-...)
Affinity DataIC50:  0.200nMAssay Description:Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM141345(US8916594, I-018)
Affinity DataIC50:  0.200nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50394224(CHEMBL2159167)
Affinity DataIC50:  0.210nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM141349(US8916594, I-029)
Affinity DataIC50:  0.220nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM141344(US8916594, I-017)
Affinity DataIC50:  0.220nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50111656(1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl)-acetyl]-pi...)
Affinity DataIC50:  0.230nMAssay Description:Tested for the inhibition of [125I]-PYY binding to HEK 293 cells stably expressed with human neuropeptide NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM141351(US8916594, I-053)
Affinity DataIC50:  0.230nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM118179(US8653125, Ia-40)
Affinity DataIC50:  0.260nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding mouse NPY Y5 receptor (Biochem. Biophys. Acta 1328: 83-89, 1997) was cloned in the expression vector (pME18S, Takebe et al. Mo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50394211(CHEMBL2159165)
Affinity DataIC50:  0.280nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50390228(CHEMBL2070161)
Affinity DataIC50:  0.290nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50394221(CHEMBL2159158)
Affinity DataIC50:  0.290nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50093646(6-Benzofuran-2-yl-2-methyl-4-piperidin-1-yl-5H-pyr...)
Affinity DataIC50:  0.300nMAssay Description:Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50093696(6-(3-Fluoro-phenyl)-2-methyl-4-piperidin-1-yl-5H-p...)
Affinity DataIC50:  0.300nMAssay Description:Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50093664(6-(4-Fluoro-phenyl)-2-methyl-4-piperidin-1-yl-5H-p...)
Affinity DataIC50:  0.300nMAssay Description:Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50390232(CHEMBL2070157)
Affinity DataIC50:  0.310nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM141342(US8916594, I-006)
Affinity DataIC50:  0.320nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM141343(US8916594, I-011)
Affinity DataIC50:  0.340nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50093691(4-(3,6-Dihydro-2H-pyridin-1-yl)-2-methyl-6-phenyl-...)
Affinity DataIC50:  0.400nMAssay Description:Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50093675(6-(3,5-Difluoro-phenyl)-2-methyl-4-piperidin-1-yl-...)
Affinity DataIC50:  0.400nMAssay Description:Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM118190(US8653125, Ic-16)
Affinity DataIC50:  0.410nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding mouse NPY Y5 receptor (Biochem. Biophys. Acta 1328: 83-89, 1997) was cloned in the expression vector (pME18S, Takebe et al. Mo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50394214(CHEMBL2159162)
Affinity DataIC50:  0.430nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50390225(CHEMBL2070140)
Affinity DataIC50:  0.430nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50394214(CHEMBL2159162)
Affinity DataIC50:  0.430nMAssay Description:Displacement of [125I]PYY from mouse NPY-Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50390222(CHEMBL2070137)
Affinity DataIC50:  0.460nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50073048(2-[4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperi...)
Affinity DataIC50:  0.470nMAssay Description:Binding affinity of the compound against human Neuropeptide Y receptor type 5 in HEK 293 cell line by using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50073048(2-[4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperi...)
Affinity DataIC50:  0.470nMAssay Description:The compound was tested for the binding affinity against Neuropeptide Y receptor type 5 in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM141357(US8916594, I-138)
Affinity DataIC50:  0.5nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50101571(1-Methyl-1-(1-methyl-2-pyridin-4-yl-ethyl)-3-(4-ph...)
Affinity DataIC50:  0.5nMAssay Description:Inhibitory activity tested against Human Neuropeptide Y5 Receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50093697(2-Methyl-4-piperidin-1-yl-6-p-tolyl-5H-pyrrolo[3,2...)
Affinity DataIC50:  0.5nMAssay Description:Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50093647(2-Methyl-6-(5-methyl-furan-2-yl)-4-piperidin-1-yl-...)
Affinity DataIC50:  0.5nMAssay Description:Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]-PYY binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50110571(CHEMBL167991 | FR-230481 | Naphthalene-1-sulfonic ...)
Affinity DataIC50:  0.540nMAssay Description:Inhibition of 125 I-PYY binding to human Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50390220(CHEMBL2070147)
Affinity DataIC50:  0.540nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50390234(CHEMBL2070155)
Affinity DataIC50:  0.550nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM118188(US8653125, Ic-13)
Affinity DataIC50:  0.560nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding mouse NPY Y5 receptor (Biochem. Biophys. Acta 1328: 83-89, 1997) was cloned in the expression vector (pME18S, Takebe et al. Mo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50258232(1-(Methylsulfonyl)-N-(5-phenylpyrimidin-2-yl)-1,2-...)
Affinity DataIC50:  0.570nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50258232(1-(Methylsulfonyl)-N-(5-phenylpyrimidin-2-yl)-1,2-...)
Affinity DataIC50:  0.570nMAssay Description:Binding affinity to human neuropeptide Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM118192(US8653125, Id-8)
Affinity DataIC50:  0.580nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding mouse NPY Y5 receptor (Biochem. Biophys. Acta 1328: 83-89, 1997) was cloned in the expression vector (pME18S, Takebe et al. Mo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50111645(1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl)-acetyl]-pi...)
Affinity DataIC50:  0.590nMAssay Description:Inhibitory concentration of total specific binding of [125I]- -PYY to HEK 293 cells transfected with Human NPY-Y5 cDNA (compound prepared by manual s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50111644(1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl)-acetyl]-pi...)
Affinity DataIC50:  0.590nMAssay Description:Inhibitory concentration of total specific binding of [125I]- -PYY to HEK 293 cells transfected with the Human NPY-Y5 cDNA (compound prepared by para...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50354066(CHEMBL1836324)
Affinity DataIC50:  0.600nMAssay Description:Antagonist activity at human NPY5 receptor assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50089055(CHEMBL273811 | N*2*-(4-Ethanesulfonylmethyl-phenyl...)
Affinity DataIC50:  0.600nMAssay Description:Antagonistic activity against neuropeptide Y receptor type 5 subtype stably expressed in LM(tk-)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM50394218(CHEMBL2159156)
Affinity DataIC50:  0.600nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Mus musculus (Mouse))
Shionogi

US Patent
LigandPNGBDBM141361(US8916594, I-147)
Affinity DataIC50:  0.610nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301643(CHEMBL570633 | trans-3'-oxo-N-(5-phenylpyrimidin-2...)
Affinity DataIC50:  0.640nMAssay Description:Displacement of [125I]PYY from human recombinant NPY Y5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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