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Found 420 Enz. Inhib. hit(s) with Target = 'Acetylcholine receptor'
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit delta(Torpedo californica)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.100nMAssay Description:Agonist activity against Nicotinic acetylcholine receptor (nAchR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487234(CHEMBL1391421)
Affinity DataKi:  0.120nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50251868((Z)-thiacloprid | CHEMBL451432 | {(2Z)-3-[(6-chlor...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  2.70nMAssay Description:Binding potency for Nicotinic acetylcholine receptor alpha-7 (rat brain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataKi:  3nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Wuhan Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50516992(CHEMBL4473371)
Affinity DataKi:  3.10nMAssay Description:Inhibition of AChE (unknown origin) by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  3.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  4.70nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  5.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  5.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  5.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  5.70nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  5.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  5.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  6.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  6.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  6.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  6.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50486223(CHEBI:39164 | acetamiprid)
Affinity DataKi:  7.20nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  11.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50038413(CHEMBL136284 | N,N'-(2,3-dihydroxylbenzyl)-N,N,N',...)
Affinity DataKi:  18nMAssay Description:Binding affinity against nicotinic acetylcholine receptor (nAChR)Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Wuhan Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50596341(CHEMBL5176418)
Affinity DataKi:  120nMAssay Description:Mixed type inhibition of AChE (unknown origin) assessed as inhibitory constant by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50472282(descyanothiacloprid)
Affinity DataKi:  130nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit epsilon(Homo sapiens (Human))
Wuhan Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataKi:  152nMAssay Description:Inhibition of AChE (unknown origin) by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50143282((-)-cytisine | (1R,5S)-1,2,3,4,5,6-Hexahydro-1,5-m...)
Affinity DataKi:  250nMAssay Description:Inhibition of [125I]alpha-bungarotoxin binding to nicotinic acetylcholine receptor alpha1 beta gamma delta of electroplaxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  290nMAssay Description:Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha/Neuronal acetylcholine receptor subunit beta-2(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50006615(CHEMBL3235483)
Affinity DataKi:  292nMAssay Description:Displacement of [3H]epibatidine from alpha2beta2-nAChR (unknown origin) expressed in HEK293 cells after 2 hrs by liquid scintillation counting analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50061562((12R,13aR)-12-Methoxy-1,4,5,6,9,11,12,13-octahydro...)
Affinity DataKi:  314nMAssay Description:Affinity for Nicotinic acetylcholine receptor alpha4-beta2 in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049750((S)-3-(azetidin-2-ylmethoxy)pyridine | 3-((S)-1-Az...)
Affinity DataKi:  314nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha(Torpedo californica)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049750((S)-3-(azetidin-2-ylmethoxy)pyridine | 3-((S)-1-Az...)
Affinity DataKi:  314nMAssay Description:Compound was evaluated for its ability to displace [125 I]alpha-bungarotoxin (alpha-BgT) from torpedo alpha1-beta1-gamma1 electroplaxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50220046(CHEMBL382243 | trimethyl({20-[(trimethylazaniumyl)...)
Affinity DataKi:  331nMAssay Description:Displacement of (+/-)-[3H]epibatidine from muscle type nAChR of Torpedo californica in hepes bufferMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  333nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50166909(10-Aza-tricyclo[6.3.1.0*2,7*]dodeca-2(7),3,5-trien...)
Affinity DataKi:  370nMAssay Description:Inhibition of [125I]alpha-bungarotoxin binding to nicotinic acetylcholine receptor alpha1 beta gamma delta of electroplaxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha(Torpedo californica)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049753(3-((R)-1-Azetidin-2-ylmethoxy)-pyridine | 3-((S)-1...)
Affinity DataKi:  384nMAssay Description:Compound was evaluated for its ability to displace [125 I]alpha-bungarotoxin (alpha-BgT) from torpedo alpha1-beta1-gamma1 electroplaxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049750((S)-3-(azetidin-2-ylmethoxy)pyridine | 3-((S)-1-Az...)
Affinity DataKi:  384nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  483nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  505nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholine receptor subunit alpha(MOUSE)
University Of Colorado

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  522nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
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