Compile Data Set for Download or QSAR
maximum 50k data
Found 80 Enz. Inhib. hit(s) with all data for entry = 2988
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387701(2-(4-(tert-butyl)piperidin-1-yl)-N-(2-(cyclopropan...)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387702(N-(2-(cyclopropanecarbonyl)-1H-indol-3-yl)-2-(8-az...)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387703(US10294214, Example 3 | methyl 3-(2-(4-cyclohexylp...)
Affinity DataEC50:  200nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387704(US10294214, Example 4)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387705(US10294214, Example 5)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387706(US10294214, Example 6)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387707(US10294214, Example 7)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387708(US10294214, Example 8)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387709(US10294214, Example 9)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387710(US10294214, Example 10)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387711(US10294214, Example 11)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387712(US10294214, Example 12)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387713(US10294214, Example 13)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387714(US10294214, Example 14)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387715(US10294214, Example 15)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387716(US10294214, Example 16)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387717(US10294214, Example 17)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387718(US10294214, Example 18)
Affinity DataEC50:  794nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387719(US10294214, Example 19)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387720(US10294214, Example 20)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387721(US10294214, Example 21)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387722(US10294214, Example 22)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387723(US10294214, Example 23)
Affinity DataEC50:  794nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387724(US10294214, Example 24)
Affinity DataEC50:  1.00E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387725(US10294214, Example 25)
Affinity DataEC50:  1.00E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387726(US10294214, Example 26)
Affinity DataEC50:  1.00E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387727(US10294214, Example 27)
Affinity DataEC50:  1.26E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387728(US10294214, Example 28)
Affinity DataEC50:  1.59E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387729(US10294214, Example 29)
Affinity DataEC50:  1.26E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387730(US10294214, Example 30)
Affinity DataEC50:  1.26E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387731(US10294214, Example 31)
Affinity DataEC50:  1.59E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387732(US10294214, Example 32)
Affinity DataEC50:  1.59E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387733(US10294214, Example 33)
Affinity DataEC50:  2.51E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387734(US10294214, Example 34)
Affinity DataEC50:  2.00E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387735(US10294214, Example 35)
Affinity DataEC50:  1.59E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387736(US10294214, Example 36)
Affinity DataEC50:  1.59E+3nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387737(US10294214, Example 37)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387738(US10294214, Example 38)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387739(US10294214, Example 39)
Affinity DataEC50:  251nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387740(US10294214, Example 40)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387741(US10294214, Example 41)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387742(US10294214, Example 42)
Affinity DataEC50:  316nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387743(US10294214, Example 43)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387744(US10294214, Example 44)
Affinity DataEC50:  398nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387745(US10294214, Example 45)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387746(US10294214, Example 46)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387747(US10294214, Example 47)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387748(US10294214, Example 48)
Affinity DataEC50:  501nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387749(US10294214, Example 49)
Affinity DataEC50:  631nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM387750(US10294214, Example 50)
Affinity DataEC50:  794nMAssay Description:Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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