Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 5905
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Court Of The University Of Dundee

US Patent
LigandPNGBDBM99922(CHEMBL1945132 | US8501991, 6)
Affinity DataIC50:  1.60E+4nMAssay Description:SIRT1 inhibition assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Court Of The University Of Dundee

US Patent
LigandPNGBDBM99917(4-tert-butyl-N-(4-(5-(dimethylamino)pentanamido)ph...)
Affinity DataIC50:  2.10E+4nMAssay Description:SIRT1 inhibition assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Court Of The University Of Dundee

US Patent
LigandPNGBDBM99920(CHEMBL1945133 | US8501991, 7)
Affinity DataIC50:  2.50E+4nMAssay Description:SIRT1 inhibition assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Court Of The University Of Dundee

US Patent
LigandPNGBDBM99918(CHEMBL1945672 | US8501991, 24)
Affinity DataIC50:  2.90E+4nMAssay Description:SIRT1 inhibition assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Court Of The University Of Dundee

US Patent
LigandPNGBDBM99919(US8501991, 5)
Affinity DataIC50:  3.20E+4nMAssay Description:SIRT1 inhibition assay.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Court Of The University Of Dundee

US Patent
LigandPNGBDBM99921(CHEMBL1945134 | US8501991, 8)
Affinity DataIC50: >6.00E+4nMAssay Description:SIRT1 inhibition assay.More data for this Ligand-Target Pair
In DepthDetails US Patent