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Found 2 Enz. Inhib. hit(s) with all data for entry = 8264
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM50401614(CHEMBL2203843 | US9403797, PAPC-A-01)
Affinity DataIC50:  6nMpH: 7.4 T: 2°CAssay Description:In vitro CHK2 kinase activity was measured in a DELFIA® assay that monitors phosphorylation of a CDC25C peptide using a specific phospho antibody...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM50401617(CHEMBL2204592 | US9403797, PAPC-A-02)
Affinity DataIC50:  8nMpH: 7.4 T: 2°CAssay Description:In vitro CHK2 kinase activity was measured in a DELFIA® assay that monitors phosphorylation of a CDC25C peptide using a specific phospho antibody...More data for this Ligand-Target Pair
In DepthDetails US Patent