Compile Data Set for Download or QSAR
maximum 50k data
Found 44 Enz. Inhib. hit(s) with all data for entry = 1474
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325586(6-Chloro-8-{5-[1-(tetrahydro-pyran-4-ylmethyl)-pip...)
Affinity DataEC50:  18nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325585(6-Chloro-8-{5-[1-(tetrahydro-pyran-4-yl)-piperidin...)
Affinity DataEC50:  5.70nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325588(5-Chloro-7-[5-(1-cyclobutyl-piperidin-4-yl)-[1,3,4...)
Affinity DataEC50:  10nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325589(6-Chloro-8-[5-(1-cyclopropyl-piperidin-4-yl)-[1,3,...)
Affinity DataEC50:  21.5nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325590(6-Chloro-8-{5-[1-(tetrahydro-pyran-4-yl)-piperidin...)
Affinity DataEC50:  7.30nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325591(6-Chloro-8-{5-[1-(3-methoxy-propyl)-piperidin-4-yl...)
Affinity DataEC50:  16.9nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325592(5-Chloro-7-{5-[1-(tetrahydro-pyran-4-ylmethyl)-pip...)
Affinity DataEC50:  21nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325593(4-[5-(4-Amino-5-chloro-2,3-dihydro-benzofuran-7-yl...)
Affinity DataEC50:  5nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325594(3-[5-(1-Cyclobutylmethyl-piperidin-4-yl)-[1,3,4]ox...)
Affinity DataEC50:  169nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325595(1-Isopropyl-3-{5-[1-(2-methoxy-ethyl)-piperidin-4-...)
Affinity DataEC50:  143nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325596(3-[5-(1-Cyclobutyl-piperidin-4-yl)-[1,3,4]oxadiazo...)
Affinity DataEC50:  127nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325597(1-Isopropyl-3-[5-(1-isopropyl-piperidin-4-yl)-[1,3...)
Affinity DataEC50:  23nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325598(3-[5-(1-Cyclopropylmethyl-piperidin-4-yl)-[1,3,4]o...)
Affinity DataEC50:  66nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325599(1-Isopropyl-3-{5-[1-(3-methyl-butyl)-piperidin-4-y...)
Affinity DataEC50:  116nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325600(3-[5-(1-Cyclopropyl-piperidin-4-yl)-[1,3,4]oxadiaz...)
Affinity DataEC50:  199nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325601(3-[5-(1-Cyclopentyl-piperidin-4-yl)-[1,3,4]oxadiaz...)
Affinity DataEC50:  72nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325602(1-Isopropyl-3-{5-[1-(tetrahydro-pyran-4-ylmethyl)-...)
Affinity DataEC50:  84.5nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325603(1-Isopropyl-3-{5-[1-(tetrahydro-pyran-4-yl)-piperi...)
Affinity DataEC50:  54nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325604(1-Isopropyl-3-[5-(2-piperidin-1-yl-ethyl)-[1,3,4]o...)
Affinity DataEC50:  181nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325557(6-chloro-8-[5-(1-cyclopropyl piperidin-4-yl)-[1,3,...)
Affinity DataEC50:  28.5nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325559(6-Chloro-8-[5-(1-cyclobutyl piperidin-4-ylmethyl)-...)
Affinity DataEC50:  47nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325559(6-Chloro-8-[5-(1-cyclobutyl piperidin-4-ylmethyl)-...)
Affinity DataEC50:  27.5nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325561(1-Isopropyl-3-{5-[1-(3-methoxy propyl) piperidin-4...)
Affinity DataEC50:  38nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325563(3-[5-(1-Cyclobutyl-piperidin-4-yl methyl)-[1,3,4]o...)
Affinity DataEC50:  18nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325564(6-Chloro-8-[5-(3-cyclobutyl-3-aza bicyclo[3.1.0]he...)
Affinity DataEC50:  4.20nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325565(5-Chloro-7-{5-[1-(tetrahydro pyran-4-yl) piperidin...)
Affinity DataEC50:  7nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325566(6-Chloro-8-{5-[1-(2-methoxy-ethyl)-piperidin-4-yl]...)
Affinity DataEC50:  15.6nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325567(6-Chloro-8-{5-[1-(3-methyl-butyl)-piperidin-4-yl]-...)
Affinity DataEC50:  2.40nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325568(6-Chloro-8-[5-(1-cyclobutylmethyl-piperidin-4-yl)-...)
Affinity DataEC50:  5.70nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325571(6-Chloro-8-[5-(1-cyclopropylmethyl-piperidin-4-yl)...)
Affinity DataEC50:  10.2nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325572(6-Chloro-8-[5-(1-isopropyl-piperidin-4-yl)-[1,3,4]...)
Affinity DataEC50:  15.3nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325573(6-Chloro-8-{5-[1-(3-methoxy-propyl)-piperidin-4-yl...)
Affinity DataEC50:  20.4nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325574(6-Chloro-8-[5-(1-cyclobutyl-piperidin-4-yl)-[1,3,4...)
Affinity DataEC50:  1.30nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325575(6-Chloro-8-[5-(1-cyclobutylmethyl-piperidin-4-yl)-...)
Affinity DataEC50:  6.20nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325576(6-Chloro-8-[5-(1-cyclobutyl-piperidin-4-yl)-[1,3,4...)
Affinity DataEC50:  13.3nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325577(6-Chloro-8-[5-(1-cyclopentyl-piperidin-4-yl)-[1,3,...)
Affinity DataEC50:  2.30nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325578(6-Chloro-8-[5-(2-piperidin-1-yl-ethyl)-[1,3,4]oxad...)
Affinity DataEC50:  53nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325579(4-[5-(5-Amino-6-chloro-chroman-8-yl)-[1,3,4]oxadia...)
Affinity DataEC50:  6.80nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325580(6-Chloro-8-[5-(3-piperidin-1-yl-propyl)-[1,3,4]oxa...)
Affinity DataEC50:  104nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325581(6-Chloro-8-[5-(1-cyclopentyl-piperidin-4-ylmethyl)...)
Affinity DataEC50:  71.2nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325582(6-Chloro-8-[5-(3-isopropyl-3-aza-bicyclo[3.1.0]hex...)
Affinity DataEC50:  48nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325583(6-Chloro-8-[5-(3-cyclobutylmethyl-3-aza-bicyclo[3....)
Affinity DataEC50:  20nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325584(6-Chloro-8-[5-(3-cyclopropylmethyl-3-aza-bicyclo[3...)
Affinity DataEC50:  25nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM325587(5-Chloro-7-[5-(1-cyclopropyl-piperidin-4-yl)-[1,3,...)
Affinity DataEC50:  60nMAssay Description:A stable CHO cell line expressing recombinant human 5-HT4 receptor and pCRE-Luc reporter system was used for cell-based assay. The assay offers a non...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent