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Found 4 Enz. Inhib. hit(s) with all data for entry = 621
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

US Patent
LigandPNGBDBM282779((S)-6-((2-oxopyrrolidin-3- yl)amino)-2-(spiro[inde...)
Affinity DataIC50:  1.30E+3nMpH: 7.3Assay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

US Patent
LigandPNGBDBM282780((S)-2-(3-oxo-3H-spiro [isobenzofuran-1,4'-piperidi...)
Affinity DataIC50:  3.86E+3nMpH: 7.3Assay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

US Patent
LigandPNGBDBM282776((S)-6-((2-oxopyrrolidin-3-yl)amino)- 2-(3H-spiro[i...)
Affinity DataIC50:  3.92E+3nMpH: 7.3Assay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

US Patent
LigandPNGBDBM282781((S)-2-(4-oxo-1-phenyl-1,3,8- triazaspiro[4.5]decan...)
Affinity DataIC50: >2.00E+4nMpH: 7.3Assay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent