Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) for PDB: 3OMP
TargetEstrogen receptor beta(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50341441(2,2,2-Trifluoro-1-(7-hydroxy-3,4-dihydroisoquinoli...)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity at human N-terminal His6-tagged ERbeta receptor LBD expressed in Escherichia coli BL21 (DE3) assessed as induction of SRC1 peptide r...More data for this Ligand-Target Pair