Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50010734
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098121(6-Methoxymethyl-3a,5b-dimethyl-3,8,11-trioxo-2,3,3...)
Affinity DataIC50:  20nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098124(CHEMBL173055 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098117(CHEMBL366754 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098120(CHEMBL263287 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098118((2S,4R)-4-Mercapto-2-(2,4,5-trifluoro-benzyloxymet...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098115(CHEMBL262054 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of DNA dependent protein kinase with hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098125(CHEMBL355195 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098115(CHEMBL262054 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098119(CHEMBL422731 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataIC50:  1.22E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098114(CHEMBL366755 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098123(CHEMBL366637 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataIC50:  1.39E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098116(CHEMBL173928 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098122(CHEMBL424579 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM15359((4E,6Z,8S,9S,10E,12S,13R,14S,16R)-13-hydroxy-8,14-...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of DNA dependent protein kinase activity without hsp90 alpha proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098124(CHEMBL173055 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataEC50:  2.80E+4nMAssay Description:Competitive binding towards Heat shock protein HSP 90-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098115(CHEMBL262054 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataEC50:  2.50E+3nMAssay Description:Competitive binding towards Heat shock protein HSP 90-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098125(CHEMBL355195 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataEC50:  4.00E+3nMAssay Description:Competitive binding towards Heat shock protein HSP 90-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098123(CHEMBL366637 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataEC50:  1.00E+4nMAssay Description:Competitive binding towards Heat shock protein HSP 90-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098118((2S,4R)-4-Mercapto-2-(2,4,5-trifluoro-benzyloxymet...)
Affinity DataEC50: >5.00E+4nMAssay Description:Competitive binding towards Heat shock protein HSP 90-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098117(CHEMBL366754 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataEC50:  7.00E+3nMAssay Description:Competitive binding towards Heat shock protein HSP 90-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098119(CHEMBL422731 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataEC50: >5.00E+4nMAssay Description:Competitive binding towards Heat shock protein HSP 90-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098121(6-Methoxymethyl-3a,5b-dimethyl-3,8,11-trioxo-2,3,3...)
Affinity DataEC50: >5.00E+4nMAssay Description:Competitive binding towards Heat shock protein HSP 90-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098122(CHEMBL424579 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataEC50:  1.60E+4nMAssay Description:Competitive binding towards Heat shock protein HSP 90-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098120(CHEMBL263287 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataEC50:  4.60E+4nMAssay Description:Competitive binding towards Heat shock protein HSP 90-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM15359((4E,6Z,8S,9S,10E,12S,13R,14S,16R)-13-hydroxy-8,14-...)
Affinity DataEC50:  1.00E+3nMAssay Description:Competitive binding towards Heat shock protein HSP 90-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098116(CHEMBL173928 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataEC50:  2.60E+4nMAssay Description:Competitive binding towards Heat shock protein HSP 90-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Department Of Molecular Oncogenesis

Curated by ChEMBL
LigandPNGBDBM50098114(CHEMBL366755 | Carbamic acid 13-hydroxy-8,14-dimet...)
Affinity DataEC50: >5.00E+4nMAssay Description:Competitive binding towards Heat shock protein HSP 90-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed