Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50042223
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422383(CHEMBL1203235)
Affinity DataIC50:  3.20nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422380(CHEMBL1203232)
Affinity DataIC50:  4.60nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422382(CHEMBL1203233)
Affinity DataIC50:  8.90nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422381(CHEMBL384790)
Affinity DataIC50:  25nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422379(CHEMBL263289)
Affinity DataIC50:  27nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422380(CHEMBL1203232)
Affinity DataIC50:  46nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422384(CHEMBL216443)
Affinity DataIC50:  81nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422380(CHEMBL1203232)
Affinity DataIC50:  1.74E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422382(CHEMBL1203233)
Affinity DataIC50:  1.86E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422382(CHEMBL1203233)
Affinity DataIC50:  1.86E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422381(CHEMBL384790)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422383(CHEMBL1203235)
Affinity DataIC50:  2.14E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422384(CHEMBL216443)
Affinity DataIC50:  3.89E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422383(CHEMBL1203235)
Affinity DataIC50:  4.68E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422378(CHEMBL122621)
Affinity DataIC50:  5.01E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422379(CHEMBL263289)
Affinity DataIC50:  5.01E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422379(CHEMBL263289)
Affinity DataIC50:  5.13E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422378(CHEMBL122621)
Affinity DataIC50:  1.62E+4nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422381(CHEMBL384790)
Affinity DataIC50:  4.17E+4nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422384(CHEMBL216443)
Affinity DataIC50:  5.50E+4nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422378(CHEMBL122621)
Affinity DataIC50:  6.76E+4nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed