Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50011280
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50101321(CHEMBL299750 | [(S)-1-((S)-1-Benzyl-2-benzyloxycar...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104576(CHEMBL89668 | [(S)-1-((S)-1-Benzyl-2-methoxycarbam...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104586(CHEMBL316418 | [(R)-1-((S)-1-Benzyl-2-benzyloxycar...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104587(CHEMBL89771 | [(S)-1-((S)-1-Benzyl-2-oxo-2-pentafl...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104579(CHEMBL313895 | {(S)-1-[(S)-1-((S)-1-Benzyl-2-benzy...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50101317(CHEMBL301598 | [(S)-1-((S)-1-Benzyl-2-ethoxycarbam...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104585(CHEMBL316135 | {(S)-1-[(S)-1-((S)-1-Benzyl-2-metho...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104577(CHEMBL419311 | {(S)-1-[(S)-1-Benzyl-2-(4-methyl-cy...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104581(CHEMBL85296 | [(S)-1-((S)-1-Benzyloxyaminooxalyl-p...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104584(CHEMBL441262 | [(S)-1-((S)-1-Benzyl-2-tert-butoxyc...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104583((S)-N-Benzyloxy-3-((R)-3-benzyloxy-2-methanesulfon...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104582((R)-N-((S)-1-Benzylcarbamoyl-2-phenyl-ethyl)-3-ben...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104578((R)-3-Benzyloxy-N-((S)-1-ethylcarbamoyl-2-phenyl-e...)
Affinity DataIC50:  56nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104580((S)-3-((R)-3-Benzyloxy-2-methanesulfonylamino-prop...)
Affinity DataIC50:  56nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104589((S)-N-Benzyloxy-3-((R)-3-benzyloxy-2-methanesulfon...)
Affinity DataIC50:  152nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104588(CHEMBL315578 | N-[(S)-1-((S)-1-Ethoxyaminooxalyl-p...)
Affinity DataIC50:  193nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed