Compile Data Set for Download or QSAR
maximum 50k data
Found 78 Enz. Inhib. hit(s) with all data for entry = 50037048
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116502(CHEMBL407428 | [22-Amino-4-carbamoyl-19-(4-hydroxy...)
Affinity DataIC50:  9nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116474(4-(2-{[22-Amino-13-carboxymethyl-19-(3-guanidino-p...)
Affinity DataIC50:  30nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116479(CHEMBL331024 | [22-Amino-19-benzyl-4-carbamoyl-10-...)
Affinity DataIC50:  50nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116506(CHEMBL432452 | [22-Amino-4-(carbamoylmethyl-carbam...)
Affinity DataIC50:  110nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116476(CHEMBL324934 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  120nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116494(22-Amino-13-carboxymethyl-19-(3-guanidino-propyl)-...)
Affinity DataIC50:  130nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116502(CHEMBL407428 | [22-Amino-4-carbamoyl-19-(4-hydroxy...)
Affinity DataIC50:  130nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116471(CHEMBL420868 | [22-Amino-4-carbamoyl-10-(1-hydroxy...)
Affinity DataIC50:  160nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116477(CHEMBL384184 | MDc(CRSDTLC)GE-NH2)
Affinity DataIC50:  190nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116487(CHEMBL325167 | [22-Amino-19-(4-amino-butyl)-4-carb...)
Affinity DataIC50:  250nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116498(CHEMBL384511 | DCRSDTLCGE-NH2)
Affinity DataIC50:  260nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116483(CHEMBL333218 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  290nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116504(CHEMBL214970 | MDc(CRSDTLC)G-NH2)
Affinity DataIC50:  340nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116484(CHEMBL117958 | [22-Amino-4-carbamoyl-10-(1-hydroxy...)
Affinity DataIC50:  390nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116494(22-Amino-13-carboxymethyl-19-(3-guanidino-propyl)-...)
Affinity DataIC50:  400nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116471(CHEMBL420868 | [22-Amino-4-carbamoyl-10-(1-hydroxy...)
Affinity DataIC50:  430nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116492(3-Amino-N-[4-carbamoyl-13-carboxymethyl-19-(3-guan...)
Affinity DataIC50:  520nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116479(CHEMBL331024 | [22-Amino-19-benzyl-4-carbamoyl-10-...)
Affinity DataIC50:  550nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116490(3-(2-Amino-4-methylsulfanyl-butyrylamino)-N-[4-car...)
Affinity DataIC50:  640nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116505(CHEMBL115901 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  800nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116488(CHEMBL116567 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  840nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116474(4-(2-{[22-Amino-13-carboxymethyl-19-(3-guanidino-p...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to block the alphaV-beta3 integrin binding to vitronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116474(4-(2-{[22-Amino-13-carboxymethyl-19-(3-guanidino-p...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116484(CHEMBL117958 | [22-Amino-4-carbamoyl-10-(1-hydroxy...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116486(CHEMBL406288 | [22-Amino-4-carbamoyl-10-(1-hydroxy...)
Affinity DataIC50:  1.10E+3nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116507(CHEMBL117435 | [22-Amino-16-sec-butyl-4-carbamoyl-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116499(AC-WERWLMDc(CRSDTLC)GESHQE-NH2 | CHEMBL439704)
Affinity DataIC50:  1.30E+3nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116487(CHEMBL325167 | [22-Amino-19-(4-amino-butyl)-4-carb...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116503(CHEMBL325039 | [22-Amino-7-sec-butyl-4-carbamoyl-1...)
Affinity DataIC50:  1.80E+3nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116505(CHEMBL115901 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  1.90E+3nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116497(CHEMBL117436 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  2.10E+3nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116473(CHEMBL443276 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  2.20E+3nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116481(22-Amino-13-carbamoylmethyl-19-(3-guanidino-propyl...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116480(CHEMBL420130 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  2.20E+3nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116486(CHEMBL406288 | [22-Amino-4-carbamoyl-10-(1-hydroxy...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116495(3-[22-Amino-4-carbamoyl-19-(3-guanidino-propyl)-10...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116480(CHEMBL420130 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116473(CHEMBL443276 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116506(CHEMBL432452 | [22-Amino-4-(carbamoylmethyl-carbam...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116477(CHEMBL384184 | MDc(CRSDTLC)GE-NH2)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116476(CHEMBL324934 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116496(CHEMBL326055 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  4.50E+3nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116474(4-(2-{[22-Amino-13-carboxymethyl-19-(3-guanidino-p...)
Affinity DataIC50:  6.10E+3nMAssay Description:Ability to block the alpha5-beta1 integrin binding to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116497(CHEMBL117436 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50370135(CHEMBL1790853)
Affinity DataIC50:  7.90E+3nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116498(CHEMBL384511 | DCRSDTLCGE-NH2)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116492(3-Amino-N-[4-carbamoyl-13-carboxymethyl-19-(3-guan...)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116504(CHEMBL214970 | MDc(CRSDTLC)G-NH2)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116493(CHEMBL117226 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  1.00E+4nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116491(CHEMBL117072 | [22-Amino-4-carbamoyl-19-(3-guanidi...)
Affinity DataIC50:  1.10E+4nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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