Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50041056
TargetMuscarinic acetylcholine receptor M2(RAT)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  13nMAssay Description:The compound was tested in vitro for binding activity against M2 muscarinic receptor in homogenates of the brainstem of rat using [3H]quinuclidinyl b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  79nMAssay Description:The compound was tested in vitro for binding activity against M1 muscarinic receptor in homogenates of the cerebral cortex of rat using [3H]pirenzepi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50404003(CHEMBL324725)
Affinity DataKi:  398nMAssay Description:The compound was tested in vitro for binding activity against M2 muscarinic receptor in homogenates of the brainstem of rat using [3H]quinuclidinyl b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50404003(CHEMBL324725)
Affinity DataKi:  398nMAssay Description:The compound was tested in vitro for binding activity against M2 muscarinic receptor in homogenates of the brainstem of rat using [3H]quinuclidinyl b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50404003(CHEMBL324725)
Affinity DataKi:  630nMAssay Description:The compound was tested in vitro for binding activity against M1 muscarinic receptor in homogenates of the cerebral cortex of rat using [3H]pirenzepi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50404003(CHEMBL324725)
Affinity DataKi:  631nMAssay Description:The compound was tested in vitro for binding activity against M1 muscarinic receptor in homogenates of the cerebral cortex of rat using [3H]pirenzepi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50404004(CHEMBL111224)
Affinity DataKi:  794nMAssay Description:The compound was tested in vitro for binding activity against M2 muscarinic receptor in homogenates of the brainstem of rat using [3H]quinuclidinyl b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50404004(CHEMBL111224)
Affinity DataKi:  794nMAssay Description:The compound was tested in vitro for binding activity against M2 muscarinic receptor in homogenates of the brainstem of rat using [3H]quinuclidinyl b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50404004(CHEMBL111224)
Affinity DataKi:  999nMAssay Description:The compound was tested in vitro for binding activity against M1 muscarinic receptor in homogenates of the cerebral cortex of rat using [3H]pirenzepi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50404004(CHEMBL111224)
Affinity DataKi:  1.00E+3nMAssay Description:The compound was tested in vitro for binding activity against M1 muscarinic receptor in homogenates of the cerebral cortex of rat using [3H]pirenzepi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed