Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 50012872
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123637(6-benzyloxy-8-(tert-butyl)-9-flouro-12,17-dihydrox...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123639(8-(tert-butyl)-9-chloro-6,12,17-trihydroxy-16-meth...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123644(6-benzyloxy-8-(tert-butyl)-12,17-dihydroxy-16-meth...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123638(9-azido-8-(tert-butyl)-6,12,17-trihydroxy-16-methy...)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123643(6-benzyloxy-8-(tert-butyl)-9,12,17-trihydroxy-16-m...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123633(8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-9-meth...)
Affinity DataKi:  610nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50251276(BN 52021 | CHEMBL514432 | GINKOLIDE B | Gingkolide...)
Affinity DataKi:  880nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123642(8-(tert-butyl)-9-flouro-6,12,17-trihydroxy-16-meth...)
Affinity DataKi:  990nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123631(8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-9-ethy...)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123632(6-benzyloxy-8-(tert-butyl)-9,12,17-trihydroxy-16-m...)
Affinity DataKi:  1.67E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123645(CHEMBL348623 | benzyl (6R,9R,12R,16S,17R)-8-tert-b...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123635(8-(tert-butyl)-6,9,12,17-tetrahydroxy-16-methyl-(6...)
Affinity DataKi:  4.26E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123636(8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-5,15,1...)
Affinity DataKi:  7.84E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123640(8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-9-amin...)
Affinity DataKi:  8.64E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123641(8-(tert-butyl)-6,9,12,17-tetrahydroxy-16-methyl-(6...)
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed