Compile Data Set for Download or QSAR
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Found 6 Enz. Inhib. hit(s) with all data for entry = 50035373
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50127377(10-[3,9-dimethyl-8-(3-methyl-4-oxopentyl)-(9R)-1,7...)
Affinity DataIC50:  500nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50127375((E)-(R)-4-Hydroxy-2-methyl-hex-2-enedioic acid 6-{...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50366883(TAUTOMYCIN)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50127378((S)-2-Hydroxy-2-methyl-succinic acid 4-{(1R,2S,3R,...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50127376((R)-2-Hydroxy-2-methyl-succinic acid 4-{(1R,2S,3R,...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University Of California Irvine

Curated by ChEMBL
LigandPNGBDBM50127379(4-Phosphono-butyric acid (1R,2S,3R,6S,7S,10R)-10-[...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed