Compile Data Set for Download or QSAR
maximum 50k data
Found 53 Enz. Inhib. hit(s) with all data for entry = 50017493
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182855(CHEMBL381296 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  35nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182863(CHEMBL207329 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  40nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182833(CHEMBL382362 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  90nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182825(CHEMBL383129 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  96nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182846(CHEMBL208255 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  140nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182844(CHEMBL378555 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  260nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182852(CHEMBL381367 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  300nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182849(CHEMBL204418 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  320nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182859(CHEMBL207331 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  350nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182851(CHEMBL383767 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  350nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182867(CHEMBL205688 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  380nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182864(CHEMBL205861 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  540nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182861(CHEMBL205641 | N-(5-((5-(1-acetylpiperazine-4-carb...)
Affinity DataIC50:  600nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182833(CHEMBL382362 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  650nMAssay Description:Inhibition of anti-CD3 antibody-induced IL2 production in human PBMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182855(CHEMBL381296 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  700nMAssay Description:Inhibition of anti-CD3 antibody-induced IL2 production in human jurkat T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182833(CHEMBL382362 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  700nMAssay Description:Inhibition of anti-CD3 antibody-induced IL2 production in human jurkat T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182853(CHEMBL207272 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  720nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182848(CHEMBL205638 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  730nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182832(CHEMBL383455 | N-(5-(3-(1-(pyrimidin-2-yl)piperazi...)
Affinity DataIC50:  900nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182839(CHEMBL205799 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182865(CHEMBL206424 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182835(CHEMBL381107 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182836(CHEMBL204624 | N-(5-(3-(1-(2H-tetrazol-5-yl)pipera...)
Affinity DataIC50:  1.44E+3nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182866(CHEMBL208523 | N-(5-((5-(1-acetylpiperazine-4-carb...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182843(CHEMBL379281 | N-(5-((4-(1-acetylpiperazine-4-carb...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182857(CHEMBL204676 | N-(5-((4-(1-acetylpiperazine-4-carb...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182852(CHEMBL381367 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of anti-CD3 antibody-induced IL2 production in human jurkat T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182828(CHEMBL425235 | N-(5-(3-(1-acetyl-1,4-diazepane-4-c...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182842(CHEMBL205691 | N-(5-(3-(1-(2-hydroxyethyl)piperazi...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182825(CHEMBL383129 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of anti-CD3 antibody-induced IL2 production in human jurkat T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182846(CHEMBL208255 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of anti-CD3 antibody-induced IL2 production in human jurkat T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182829(CHEMBL427033 | N-(5-(4-acetamido-3-(1-acetylpipera...)
Affinity DataIC50:  2.42E+3nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182850(CHEMBL205541 | N-(5-(3-(morpholine-4-carbonyl)benz...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182862((E)-N-(5-(4-(4-acetylpiperazin-1-yl)-4-oxobut-2-en...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182840((E)-N-(5-(3-(1-acetylpiperazine-4-carbonyl)styryl)...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182849(CHEMBL204418 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of anti-CD3 antibody-induced IL2 production in human jurkat T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182860(CHEMBL207732 | N-(5-(3-(4-methylpiperidine-1-carbo...)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182856(CHEMBL205599 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182863(CHEMBL207329 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of anti-CD3 antibody-induced IL2 production in human jurkat T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182841(CHEMBL205585 | N-(5-(3-acetamido-5-(1-acetylpipera...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182845(4-(dimethylamino)-N-[5-({[3-(dimethylcarbamoyl)phe...)
Affinity DataIC50:  1.48E+4nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182827(CHEMBL440046 | N-(5-(5-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182831(CHEMBL205572 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182837(CHEMBL380075 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182854(CHEMBL205959 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182838(CHEMBL208165 | N-(5-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182824(4-(dimethylamino)-N-[5-({[3-(phenylcarbamoyl)pheny...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182868(CHEMBL208254 | N-(4-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182847(4-(dimethylamino)-N-{5-[({3-[(2-acetamidoethyl)car...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50182834(CHEMBL208265 | N-(6-(3-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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