Compile Data Set for Download or QSAR
maximum 50k data
Found 48 Enz. Inhib. hit(s) with all data for entry = 50018175
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192297(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  500nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192291(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  500nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50100110(1-[4-Amino-9-(tert-butyl-dimethyl-silanyloxy)-6-(t...)
Affinity DataIC50:  700nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50175613(1-[4-Amino-9-(tert-butyl-dimethyl-silanyloxy)-6-(t...)
Affinity DataIC50:  800nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50169035(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50106919(CHEMBL105018 | {3-[3-(tert-Butyl-dimethyl-silanylo...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192289(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50100110(1-[4-Amino-9-(tert-butyl-dimethyl-silanyloxy)-6-(t...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192302(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50175617(2-{3-[4-Amino-9-(tert-butyl-dimethyl-silanyloxy)-6...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192291(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192296(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50175613(1-[4-Amino-9-(tert-butyl-dimethyl-silanyloxy)-6-(t...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192302(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192304((S)-2-(2-{3-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-d...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50175628(BDBM50192299 | CHEMBL379599 | {3-[4-Amino-9-(tert-...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50175609(5-{3-[4-Amino-9-(tert-butyl-dimethyl-silanyloxy)-6...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192306(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192293(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192287(CHEMBL212868 | N-[(5R,6R,8R,9R)-9-(tert-butyl-dime...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192297(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192301(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192294(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192296(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50175626(BDBM50192300 | CHEMBL378474 | [(3-{3-[4-Amino-9-(t...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192290(CHEMBL379337 | N-[(5R,6R,8R,9R)-6-benzyloxymethyl-...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50175628(BDBM50192299 | CHEMBL379599 | {3-[4-Amino-9-(tert-...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50106919(CHEMBL105018 | {3-[3-(tert-Butyl-dimethyl-silanylo...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192289(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192288(3-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50024581(CHEMBL3142813)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50024581(CHEMBL3142813)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50169035(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50175609(5-{3-[4-Amino-9-(tert-butyl-dimethyl-silanyloxy)-6...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50175617(2-{3-[4-Amino-9-(tert-butyl-dimethyl-silanyloxy)-6...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192290(CHEMBL379337 | N-[(5R,6R,8R,9R)-6-benzyloxymethyl-...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192301(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192293(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192307(3-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192306(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192292((S)-2-(2-{3-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-d...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192307(3-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50175626(BDBM50192300 | CHEMBL378474 | [(3-{3-[4-Amino-9-(t...)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192288(3-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  1.17E+4nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192292((S)-2-(2-{3-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-d...)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192304((S)-2-(2-{3-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-d...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192287(CHEMBL212868 | N-[(5R,6R,8R,9R)-9-(tert-butyl-dime...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50192294(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of FLAG-p66/HIS-p51-mediated HIV1 reverse transcriptase dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed