Compile Data Set for Download or QSAR
maximum 50k data
Found 74 Enz. Inhib. hit(s) with all data for entry = 50037821
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195169(2,4-dichloro-N-((4-(morpholine-4-carbonyl)-1-(prop...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195169(2,4-dichloro-N-((4-(morpholine-4-carbonyl)-1-(prop...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of rat GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195181(2,4-dichloro-5-fluoro-N-((4-(morpholine-4-carbonyl...)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195181(2,4-dichloro-5-fluoro-N-((4-(morpholine-4-carbonyl...)
Affinity DataIC50:  7.40nMAssay Description:Inhibition of rat GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Mus musculus)
Merck And

Curated by ChEMBL
LigandPNGBDBM50195169(2,4-dichloro-N-((4-(morpholine-4-carbonyl)-1-(prop...)
Affinity DataIC50:  7.60nMAssay Description:Inhibition of mouse GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195166(3-chloro-2,6-difluoro-N-((4-(morpholine-4-carbonyl...)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195170(2-chloro-N-((4-(morpholine-4-carbonyl)-1-(propylsu...)
Affinity DataIC50:  9.70nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195173(2-chloro-4-fluoro-N-((4-(morpholine-4-carbonyl)-1-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of rat GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195178(2-chloro-6-fluoro-N-((4-(morpholine-4-carbonyl)-1-...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195173(2-chloro-4-fluoro-N-((4-(morpholine-4-carbonyl)-1-...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195170(2-chloro-N-((4-(morpholine-4-carbonyl)-1-(propylsu...)
Affinity DataIC50:  18nMAssay Description:Inhibition of rat GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Mus musculus)
Merck And

Curated by ChEMBL
LigandPNGBDBM50195181(2,4-dichloro-5-fluoro-N-((4-(morpholine-4-carbonyl...)
Affinity DataIC50:  19nMAssay Description:Inhibition of mouse GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195166(3-chloro-2,6-difluoro-N-((4-(morpholine-4-carbonyl...)
Affinity DataIC50:  20nMAssay Description:Inhibition of rat GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195178(2-chloro-6-fluoro-N-((4-(morpholine-4-carbonyl)-1-...)
Affinity DataIC50:  22nMAssay Description:Inhibition of rat GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Mus musculus)
Merck And

Curated by ChEMBL
LigandPNGBDBM50195173(2-chloro-4-fluoro-N-((4-(morpholine-4-carbonyl)-1-...)
Affinity DataIC50:  29nMAssay Description:Inhibition of mouse GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Mus musculus)
Merck And

Curated by ChEMBL
LigandPNGBDBM50195166(3-chloro-2,6-difluoro-N-((4-(morpholine-4-carbonyl...)
Affinity DataIC50:  43nMAssay Description:Inhibition of mouse GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195168(2-fluoro-N-((4-(morpholine-4-carbonyl)-1-(propylsu...)
Affinity DataIC50:  43nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Mus musculus)
Merck And

Curated by ChEMBL
LigandPNGBDBM50195178(2-chloro-6-fluoro-N-((4-(morpholine-4-carbonyl)-1-...)
Affinity DataIC50:  57nMAssay Description:Inhibition of mouse GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195167(4-fluoro-N-((4-(morpholine-4-carbonyl)-1-(propylsu...)
Affinity DataIC50:  68nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195171(4-((2,4-dichlorobenzamido)methyl)-N-((3-methyloxet...)
Affinity DataIC50:  69nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195172(CHEMBL220987 | N-((4-(morpholine-4-carbonyl)-1-(pr...)
Affinity DataIC50:  88nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Mus musculus)
Merck And

Curated by ChEMBL
LigandPNGBDBM50195170(2-chloro-N-((4-(morpholine-4-carbonyl)-1-(propylsu...)
Affinity DataIC50:  95nMAssay Description:Inhibition of mouse GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195175(CHEMBL223491 | N-((4-(3-aminoazetidine-1-carbonyl)...)
Affinity DataIC50:  109nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195179(2,6-difluoro-N-((4-(morpholine-4-carbonyl)-1-(prop...)
Affinity DataIC50:  131nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195163(4-((2,4-dichlorobenzamido)methyl)-N,N-dimethyl-1-(...)
Affinity DataIC50:  181nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195174(CHEMBL220948 | N-((4-(morpholine-4-carbonyl)-1-(pr...)
Affinity DataIC50:  264nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195165(2,4-dichloro-N-((4-(cyclopropanecarbonyl)-1-(propy...)
Affinity DataIC50:  472nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195180(4-((2,4-dichlorobenzamido)methyl)-N-ethyl-1-(propy...)
Affinity DataIC50:  517nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195183(2,4-dichloro-N-((4-(3-(dimethylamino)pyrrolidine-1...)
Affinity DataIC50:  544nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195162(2,4-dichloro-N-((4-(1-methylpiperazine-4-carbonyl)...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195182((R)-2,4-dichloro-N-(1-(4-(morpholine-4-carbonyl)-1...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195176((S)-2,4-dichloro-N-(1-(4-(morpholine-4-carbonyl)-1...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195164(CHEMBL220179 | N-((4-(morpholine-4-carbonyl)-1-(pr...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195177(CHEMBL373556 | N-((4-(morpholine-4-carbonyl)-1-(pr...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human GlyT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195171(4-((2,4-dichlorobenzamido)methyl)-N-((3-methyloxet...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195174(CHEMBL220948 | N-((4-(morpholine-4-carbonyl)-1-(pr...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195177(CHEMBL373556 | N-((4-(morpholine-4-carbonyl)-1-(pr...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195169(2,4-dichloro-N-((4-(morpholine-4-carbonyl)-1-(prop...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195178(2-chloro-6-fluoro-N-((4-(morpholine-4-carbonyl)-1-...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195166(3-chloro-2,6-difluoro-N-((4-(morpholine-4-carbonyl...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195173(2-chloro-4-fluoro-N-((4-(morpholine-4-carbonyl)-1-...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195165(2,4-dichloro-N-((4-(cyclopropanecarbonyl)-1-(propy...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195172(CHEMBL220987 | N-((4-(morpholine-4-carbonyl)-1-(pr...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195163(4-((2,4-dichlorobenzamido)methyl)-N,N-dimethyl-1-(...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195164(CHEMBL220179 | N-((4-(morpholine-4-carbonyl)-1-(pr...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195179(2,6-difluoro-N-((4-(morpholine-4-carbonyl)-1-(prop...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195162(2,4-dichloro-N-((4-(1-methylpiperazine-4-carbonyl)...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195170(2-chloro-N-((4-(morpholine-4-carbonyl)-1-(propylsu...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195181(2,4-dichloro-5-fluoro-N-((4-(morpholine-4-carbonyl...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL
LigandPNGBDBM50195167(4-fluoro-N-((4-(morpholine-4-carbonyl)-1-(propylsu...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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