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Found 35 Enz. Inhib. hit(s) with all data for entry = 50025693
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)
Affinity DataIC50:  110nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245529(CHEMBL488022 | R)-{4-[{2-[3-Amino-4-(2,4,5-trifluo...)
Affinity DataIC50:  510nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245468((R)-{4-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50:  690nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245275((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  710nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245359((R)-4-({2-[3-Amino-4-(2,4,5-trifluorophenyl)butyry...)
Affinity DataIC50:  770nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245404((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245274((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245503((R)-4-[({2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245358((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245439((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245321((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245318((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245319((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245469((R)-{3-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245438((R)-{3-[({2-[3-Amino-4-(2,4,5-trifluorophenyl)buty...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245406((R)-{4-[({2-[3-Amino-4-(2,4,5-trifluorophenyl)buty...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245556((R)-{4-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245277((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245527((R)-{4-[({2-[3-Amino-4-(2,4,5-trifluorophenyl)buty...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245501((R)-{4-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245555((R)-{4-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245276((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245528((R)-{3-[({2-[3-Amino-4-(2,4,5-trifluorophenyl)buty...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245357((R)-4-[({2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245405((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245502((R)-{4-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245403((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245553((R)-{3-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245470((R)-{2-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245320((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245526((R)-4-({2-[3-Amino-4-(2,4,5-trifluorophenyl)butyry...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245360((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245554((R)-{2-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245441((R)-4-({2-[3-Amino-4-(2,4,5-trifluorophenyl)butyry...)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50245440((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 mins by fluorometry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed