Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 50026025
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260622((S)-7-(Toluene-4-sulfonyl)-1,4-dioxa-7-aza-spiro[4...)
Affinity DataIC50:  3nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260661((S)-2-(Toluene-4-sulfonyl)-6,10-dioxa-2-aza-spiro-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260662((S)-2-(Toluene-4-sulfonyl)-6,11-dioxa-2-aza-spiro-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260663((S)-7-Benzenesulfonyl-1,4-dioxa-7-aza-spiro[4.4]-n...)
Affinity DataIC50:  8nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247539(CHEMBL472915 | N-((3S,5S)-1-((E)-3-(3,4-dimethoxyp...)
Affinity DataIC50:  9nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260664((S)-2-Benzenesulfonyl-6,10-dioxa-2-aza-spiro[4.5]-...)
Affinity DataIC50:  11nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260665((S)-2-Benzenesulfonyl-6,11-dioxa-2-aza-spiro[4.6]-...)
Affinity DataIC50:  12nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50253922(4-Hydroxy-1-(toluene-4-sulfonyl)-pyrrolidine-2-car...)
Affinity DataIC50:  100nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260537((S)-7-(Toluene-4-sulfonyl)-1,4-dioxa-7-aza-spiro[4...)
Affinity DataIC50:  100nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260619((S)-7-Benzenesulfonyl-1,4-dioxa-7-aza-spiro[4.4]no...)
Affinity DataIC50:  200nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260617((S)-2-(Toluene-4-sulfonyl)-6,10-dioxa-2-aza-spiro[...)
Affinity DataIC50:  200nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260618((S)-2-(Toluene-4-sulfonyl)-6,11-dioxa-2-aza-spiro-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260507(4-Oxo-1-(toluene-4-sulfonyl)-pyrrolidine-2-carboxy...)
Affinity DataIC50:  400nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50253923(1-Benzenesulfonyl-4-hydroxy-pyrrolidine-2-carboxyl...)
Affinity DataIC50:  800nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260620((S)-2-Benzenesulfonyl-6,10-dioxa-2-aza-spiro-[4.5]...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260621((S)-2-Benzenesulfonyl-6,11-dioxa-2-aza-spiro[4.6]-...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260508(1-Benzenesulfonyl-4-oxo-pyrrolidine-2-carboxylicac...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50253924(4-Hydroxy-1-methanesulfonyl-pyrrolidine-2-carboxyl...)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260509(1-Methanesulfonyl-4-oxo-pyrrolidine-2-carboxylicac...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50253922(4-Hydroxy-1-(toluene-4-sulfonyl)-pyrrolidine-2-car...)
Affinity DataIC50:  3.84E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50253924(4-Hydroxy-1-methanesulfonyl-pyrrolidine-2-carboxyl...)
Affinity DataIC50:  4.16E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260622((S)-7-(Toluene-4-sulfonyl)-1,4-dioxa-7-aza-spiro[4...)
Affinity DataIC50:  4.85E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50253923(1-Benzenesulfonyl-4-hydroxy-pyrrolidine-2-carboxyl...)
Affinity DataIC50:  5.38E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260507(4-Oxo-1-(toluene-4-sulfonyl)-pyrrolidine-2-carboxy...)
Affinity DataIC50:  5.49E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260663((S)-7-Benzenesulfonyl-1,4-dioxa-7-aza-spiro[4.4]-n...)
Affinity DataIC50:  5.78E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260661((S)-2-(Toluene-4-sulfonyl)-6,10-dioxa-2-aza-spiro-...)
Affinity DataIC50:  6.18E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260662((S)-2-(Toluene-4-sulfonyl)-6,11-dioxa-2-aza-spiro-...)
Affinity DataIC50:  7.32E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260508(1-Benzenesulfonyl-4-oxo-pyrrolidine-2-carboxylicac...)
Affinity DataIC50:  7.58E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260664((S)-2-Benzenesulfonyl-6,10-dioxa-2-aza-spiro[4.5]-...)
Affinity DataIC50:  8.27E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260509(1-Methanesulfonyl-4-oxo-pyrrolidine-2-carboxylicac...)
Affinity DataIC50:  9.26E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260665((S)-2-Benzenesulfonyl-6,11-dioxa-2-aza-spiro[4.6]-...)
Affinity DataIC50:  1.07E+5nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260618((S)-2-(Toluene-4-sulfonyl)-6,11-dioxa-2-aza-spiro-...)
Affinity DataIC50:  1.24E+5nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260621((S)-2-Benzenesulfonyl-6,11-dioxa-2-aza-spiro[4.6]-...)
Affinity DataIC50:  1.35E+5nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247539(CHEMBL472915 | N-((3S,5S)-1-((E)-3-(3,4-dimethoxyp...)
Affinity DataIC50:  1.42E+5nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260619((S)-7-Benzenesulfonyl-1,4-dioxa-7-aza-spiro[4.4]no...)
Affinity DataIC50:  1.51E+5nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260537((S)-7-(Toluene-4-sulfonyl)-1,4-dioxa-7-aza-spiro[4...)
Affinity DataIC50:  1.56E+5nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260620((S)-2-Benzenesulfonyl-6,10-dioxa-2-aza-spiro-[4.5]...)
Affinity DataIC50:  1.68E+5nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260617((S)-2-(Toluene-4-sulfonyl)-6,10-dioxa-2-aza-spiro[...)
Affinity DataIC50:  1.74E+5nMAssay Description:Inhibition of aminopeptidase N (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed