Affinity DataKi: 50nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 505nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.65E+3nMAssay Description:Agonist activity against human GPR109a assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 8.30E+3nMAssay Description:Agonist activity against human GPR109a assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.08E+3nMAssay Description:Agonist activity against mouse GPR109a assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.04E+4nMAssay Description:Agonist activity against human GPR109a assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Agonist activity against human GPR109a assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonist activity against mouse GPR109a assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Agonist activity against rat GPR109a assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:Agonist activity against mouse GPR109a assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 860nMAssay Description:Agonist activity against human GPR109a assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.22E+4nMAssay Description:Agonist activity against mouse GPR109a assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair