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Found 2 Enz. Inhib. hit(s) with all data for entry = 50041748
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50414756(CHEMBL569201)
Affinity DataKd:  281nMAssay Description:Antagonist activity at Alpha-1B adrenoceptor in guinea pig spleen assessed as inhibition of noradrenaline-induced contraction after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50414756(CHEMBL569201)
Affinity DataKd:  55.0nMAssay Description:Antagonist activity at Alpha-1D adrenoceptor in Wistar rat thoracic aorta assessed as inhibition of noradrenaline-induced contraction after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed