Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50030865
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303019(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50:  1.72nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303018(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50:  2.13nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303027(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50:  2.56nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303014(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50:  2.56nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303011(2-tert-butyl-5-(5-(4-chlorophenyl)-1-(2,4-dichloro...)
Affinity DataIC50:  2.83nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303022(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(5-...)
Affinity DataIC50:  3.03nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303020(2-(5-(4-chlorophenyl)-3-(5-(1-(4-chlorophenyl)cycl...)
Affinity DataIC50:  3.23nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303017(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50:  3.69nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303028(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50:  3.70nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303009(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(5-...)
Affinity DataIC50:  3.93nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303013(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(5-...)
Affinity DataIC50:  4.14nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303029(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-3-(5-(...)
Affinity DataIC50:  4.21nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303025(2-(5-(4-bromophenyl)-3-(5-(1-(4-chlorophenyl)cyclo...)
Affinity DataIC50:  4.44nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303016(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-3-(5-(...)
Affinity DataIC50:  4.70nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303026(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-3-(5-(...)
Affinity DataIC50:  4.86nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303015(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50:  4.91nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303024(2-(5-(4-bromophenyl)-3-(5-tert-butyl-1,3,4-thiadia...)
Affinity DataIC50:  4.93nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50:  5nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303008(2-tert-butyl-5-(5-(4-chlorophenyl)-1-(2,4-dichloro...)
Affinity DataIC50:  6.47nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303023(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(5-...)
Affinity DataIC50:  7.39nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303012(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(5-...)
Affinity DataIC50:  10.3nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303010(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(5-...)
Affinity DataIC50:  14.7nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303021(2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(5-...)
Affinity DataIC50:  26.9nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303019(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50:  38.5nMAssay Description:Binding affinity to human CB2 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50:  92.5nMAssay Description:Binding affinity to human CB2 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303019(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50:  245nMAssay Description:Displacement of [3H]WIN552122 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303014(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50:  414nMAssay Description:Displacement of [3H]WIN552122 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303027(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50:  427nMAssay Description:Displacement of [3H]WIN552122 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataIC50:  1.76E+3nMAssay Description:Displacement of [3H]WIN552122 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50303028(2-(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-(5-m...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]WIN552122 from human CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed