Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50039069
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378670(CHEMBL600474)
Affinity DataKi:  5.20E+4nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50109609((2R)-2-amino-3-mercaptopropanoic acid | (2R)-2-ami...)
Affinity DataKi:  5.90E+4nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378666(CHEMBL601837)
Affinity DataKi:  6.00E+4nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378667(CHEMBL604574)
Affinity DataKi:  6.40E+4nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378668(CHEMBL606915)
Affinity DataKi:  1.13E+5nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378669(CHEMBL591770)
Affinity DataKi:  1.17E+5nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378665(CHEMBL590556)
Affinity DataKi:  1.47E+5nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50109609((2R)-2-amino-3-mercaptopropanoic acid | (2R)-2-ami...)
Affinity DataIC50:  1.16E+5nMAssay Description:Inhibition of amino acid transport system xc- in human SNB19 cells assessed as [3H]L-glutamate uptake by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378666(CHEMBL601837)
Affinity DataIC50:  1.27E+5nMAssay Description:Inhibition of amino acid transport system xc- in human SNB19 cells assessed as [3H]L-glutamate uptake by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378667(CHEMBL604574)
Affinity DataIC50:  1.29E+5nMAssay Description:Inhibition of amino acid transport system xc- in human SNB19 cells assessed as [3H]L-glutamate uptake by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378668(CHEMBL606915)
Affinity DataIC50:  2.25E+5nMAssay Description:Inhibition of amino acid transport system xc- in human SNB19 cells assessed as [3H]L-glutamate uptake by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378665(CHEMBL590556)
Affinity DataIC50:  2.90E+5nMAssay Description:Inhibition of amino acid transport system xc- in human SNB19 cells assessed as [3H]L-glutamate uptake by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed