Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 50031974
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322591(3-tert-butyl-9H-carbazole | CHEMBL1170621)
Affinity DataIC50:  240nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322579(2-(trifluoromethyl)-9H-carbazole | CHEMBL1173704)
Affinity DataIC50:  260nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322580(2-tert-butyl-9H-carbazole | CHEMBL1173703)
Affinity DataIC50:  300nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322578(CHEMBL1173167 | methyl 7-tert-butyl-9H-carbazole-3...)
Affinity DataIC50:  390nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322585(2-(trifluoromethoxy)-9H-carbazole | CHEMBL1171980)
Affinity DataIC50:  510nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322584(2-(difluoromethyl)-9H-carbazole | CHEMBL1170284)
Affinity DataIC50:  870nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322575(3-(trifluoromethyl)-9H-carbazole | CHEMBL1170444)
Affinity DataIC50:  950nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322590(2-tert-butyl-7-(trifluoromethyl)-9H-carbazole | CH...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322583(2-isopropyl-9H-carbazole | CHEMBL1170460)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322598(2,3,4,11-tetrahydro-1H-benzo[a]carbazole | CHEMBL1...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322576(1-(7-methyl-9H-carbazol-3-yl)ethanone | CHEMBL1173...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322582(2-ethyl-9H-carbazole | CHEMBL1171435)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322586(2-tert-butoxy-9H-carbazole | CHEMBL1170845)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322595(1-(trifluoromethyl)-9H-carbazole | CHEMBL1169609)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322599(11H-benzo[a]carbazole | CHEMBL1173622)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322596(9-methyl-2-(trifluoromethyl)-9H-carbazole | CHEMBL...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50198301((3aS,10R)-2-butyl-10-(3-hydroxy-phenyl)-3a,4,9,10-...)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322577(6-fluoro-2-methyl-9H-carbazole | CHEMBL1172721)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322573(3-methyl-6-(trifluoromethyl)-9H-carbazole | CHEMBL...)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322574(2-methyl-6-(trifluoromethyl)-9H-carbazole | CHEMBL...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322589(7-tert-butyl-9H-carbazole-3-carboxylic acid | CHEM...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322587(CHEMBL1172394 | methyl 9H-carbazole-2-carboxylate)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322588(9H-carbazole-2-carbaldehyde | CHEMBL1172395)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322594(1-tert-butyl-9H-carbazole | CHEMBL1172393)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322592(9H-carbazole-3-carbaldehyde | CHEMBL1172392)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322581(2-methyl-9H-carbazole | CHEMBL1173640)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322593(1-methyl carbazole | 1-methyl-9H-carbazole | CHEMB...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50322597(7,8,9,10-tetrahydro-5H-benzo[b]carbazole | CHEMBL1...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human C-terminally His6-tagged microtubule-activated KSP motor domain ATPase activity after 30 mins by luciferase-derived luminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed