Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 50001117
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi:  500nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(5-(1H-Indol-3-yl)-6-piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(5-(1H-Indol-3-yl)-6-piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]-8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(3-(3-Piperidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-1...)
Affinity DataKi:  8.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(3-(3-Piperidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-1...)
Affinity DataKi:  8.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-...)
Affinity DataKi:  8.50E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(3-(3-Piperidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-1...)
Affinity DataKi:  1.35E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-...)
Affinity DataKi:  1.70E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-...)
Affinity DataKi:  1.70E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataKi:  2.30E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataKi:  2.30E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataKi:  3.20E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(5-(1H-Indol-3-yl)-6-piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataKi:  6.10E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(5-(1H-Indol-3-yl)-6-piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataKi:  6.10E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012984(5-Phenyl-6-piperidin-1-yl-bicyclo[2.2.2]octan-2-on...)
Affinity DataKi:  1.32E+5nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012984(5-Phenyl-6-piperidin-1-yl-bicyclo[2.2.2]octan-2-on...)
Affinity DataKi:  2.74E+5nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]-8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataIC50:  680nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(5-(1H-Indol-3-yl)-6-piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(5-(1H-Indol-3-yl)-6-piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(3-(3-Piperidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-1...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(3-(3-Piperidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-1...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(3-(3-Piperidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-1...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(3-(3-Piperidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-1...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]-8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-...)
Affinity DataIC50:  2.40E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]-8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]-8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-...)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]-8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]oct-5-en-2-yl)-...)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(5-(1H-Indol-3-yl)-6-piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataIC50:  8.60E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(5-(1H-Indol-3-yl)-6-piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataIC50:  8.60E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012984(5-Phenyl-6-piperidin-1-yl-bicyclo[2.2.2]octan-2-on...)
Affinity DataIC50:  1.81E+5nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012984(5-Phenyl-6-piperidin-1-yl-bicyclo[2.2.2]octan-2-on...)
Affinity DataIC50:  3.58E+5nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed