Found 73 Enz. Inhib. hit(s) with all data for entry = 50033679 
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 570nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 840nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 7.00E+3nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 7.80E+3nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+4nMAssay Description:Displacement of [3H]-MPEP from human mGluR5 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate-induced calcium mobilization aft...More data for this Ligand-Target Pair
