Compile Data Set for Download or QSAR
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Found 22 Enz. Inhib. hit(s) with all data for entry = 50034187
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358537(CHEMBL1923536)
Affinity DataEC50:  0.450nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358558(CHEMBL1923557)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358539(CHEMBL1923538)
Affinity DataEC50:  0.870nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358540(CHEMBL1923539)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358541(CHEMBL1923540)
Affinity DataEC50:  6.48nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358542(CHEMBL1923541)
Affinity DataEC50:  0.560nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358543(CHEMBL1923542)
Affinity DataEC50:  1.47nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358544(CHEMBL1923543)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358545(CHEMBL1923544)
Affinity DataEC50:  2.11nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358546(CHEMBL1923545)
Affinity DataEC50:  1.55nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358547(CHEMBL1923546)
Affinity DataEC50:  3.23nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358548(CHEMBL1923547)
Affinity DataEC50:  1.95nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358549(CHEMBL1923548)
Affinity DataEC50:  1.86nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358550(CHEMBL1923549 | US9676818, 6d)
Affinity DataEC50:  4.44nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358551(CHEMBL1923550)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358552(CHEMBL1923551)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358553(CHEMBL1923552)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358554(CHEMBL1923553)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358555(CHEMBL1923554)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358556(CHEMBL1923555)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358557(CHEMBL1923556)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50358538(CHEMBL1923537)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as NF-kappaB induction measured soluble alkaline phosphatase after 12 hrs by spectr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed