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Found 4 Enz. Inhib. hit(s) with all data for entry = 50045924
TargetSolute carrier organic anion transporter family member 1B3(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50088500(CHEBI:74023 | Dioscin)
Affinity DataKi:  1.03E+3nMAssay Description:Cellular uptake in HEK293 cells expressing OATP1B3 (unknown origin) assessed as inhibition of telmisartan-mediated drug transportMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1B3(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50088500(CHEBI:74023 | Dioscin)
Affinity DataKi:  1.43E+3nMAssay Description:Cellular uptake in HEK293 cells expressing OATP1B3 (unknown origin) assessed as inhibition of cyclosporin A-mediated drug transportMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1B3(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50088500(CHEBI:74023 | Dioscin)
Affinity DataKi:  4.55E+3nMAssay Description:Cellular uptake in HEK293 cells expressing OATP1B3 (unknown origin) assessed as inhibition of rifampicin-mediated drug transportMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1B3(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50088500(CHEBI:74023 | Dioscin)
Affinity DataKi:  8.29E+3nMAssay Description:Cellular uptake in HEK293 cells expressing OATP1B3 (unknown origin) assessed as inhibition of (-)-epigallocatechin gallate-mediated drug transportMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed