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Found 50 Enz. Inhib. hit(s) with all data for entry = 50043012
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434513(CHEMBL2385778)
Affinity DataIC50:  800nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434513(CHEMBL2385778)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434506(CHEMBL2385785)
Affinity DataIC50:  1.37E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434511(CHEMBL2385780)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  2.09E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434509(CHEMBL2385782)
Affinity DataIC50:  2.25E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434527(CHEMBL2385764)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434529(CHEMBL2385762)
Affinity DataIC50:  2.86E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434515(CHEMBL2385776)
Affinity DataIC50:  2.91E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434516(CHEMBL2385775)
Affinity DataIC50:  3.07E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434526(CHEMBL2385765)
Affinity DataIC50:  3.31E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434517(CHEMBL2385774)
Affinity DataIC50:  3.78E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434528(CHEMBL2385763)
Affinity DataIC50:  5.22E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434518(CHEMBL2385773)
Affinity DataIC50:  5.39E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434506(CHEMBL2385785)
Affinity DataIC50:  5.58E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434523(CHEMBL2385768)
Affinity DataIC50:  6.22E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434509(CHEMBL2385782)
Affinity DataIC50:  6.26E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434510(CHEMBL2385781)
Affinity DataIC50:  6.27E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434514(CHEMBL2385777)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434522(CHEMBL2385769)
Affinity DataIC50:  7.09E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434512(CHEMBL2385779)
Affinity DataIC50:  8.09E+3nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434524(CHEMBL2385767)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434525(CHEMBL2385766)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434511(CHEMBL2385780)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434518(CHEMBL2385773)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434523(CHEMBL2385768)
Affinity DataIC50:  1.59E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434521(CHEMBL2385770)
Affinity DataIC50:  1.67E+4nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434526(CHEMBL2385765)
Affinity DataIC50:  1.86E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434520(CHEMBL2385771)
Affinity DataIC50:  1.89E+4nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434517(CHEMBL2385774)
Affinity DataIC50:  1.93E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  1.93E+4nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434519(CHEMBL2385772)
Affinity DataIC50:  2.35E+4nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434527(CHEMBL2385764)
Affinity DataIC50:  2.41E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434507(CHEMBL2385784)
Affinity DataIC50:  2.63E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434524(CHEMBL2385767)
Affinity DataIC50:  2.83E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434508(CHEMBL2385783)
Affinity DataIC50:  2.88E+4nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434519(CHEMBL2385772)
Affinity DataIC50:  2.99E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434515(CHEMBL2385776)
Affinity DataIC50:  3.24E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434512(CHEMBL2385779)
Affinity DataIC50:  3.43E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434521(CHEMBL2385770)
Affinity DataIC50:  3.68E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434508(CHEMBL2385783)
Affinity DataIC50:  3.72E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434510(CHEMBL2385781)
Affinity DataIC50:  3.75E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434516(CHEMBL2385775)
Affinity DataIC50:  3.97E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434525(CHEMBL2385766)
Affinity DataIC50:  4.02E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434528(CHEMBL2385763)
Affinity DataIC50:  4.04E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434514(CHEMBL2385777)
Affinity DataIC50:  4.04E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434520(CHEMBL2385771)
Affinity DataIC50:  4.42E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434522(CHEMBL2385769)
Affinity DataIC50:  4.65E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434507(CHEMBL2385784)
Affinity DataIC50:  4.98E+4nMAssay Description:Inhibition of equine serum BuChE using S-butyrylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50434529(CHEMBL2385762)
Affinity DataIC50:  6.87E+4nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate incubated for 15 mins prior to substrate addition measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed