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Found 32 Enz. Inhib. hit(s) with all data for entry = 50043354
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439721(CHEMBL2418953)
Affinity DataIC50:  2nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439711(CHEMBL2418954)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using 1alpha-phosphotidylinositol by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439711(CHEMBL2418954)
Affinity DataIC50:  4nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439726(CHEMBL2418948)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439711(CHEMBL2418954)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of PI3Kgamma (unknown origin) using 1alpha-phosphotidylinositol by luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439723(CHEMBL2418951)
Affinity DataIC50:  14nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439722(CHEMBL2418952)
Affinity DataIC50:  25nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439713(CHEMBL2418943)
Affinity DataIC50:  33nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439714(CHEMBL2418944)
Affinity DataIC50:  36nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439727(CHEMBL2418947)
Affinity DataIC50:  54nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439728(CHEMBL2418946)
Affinity DataIC50:  68nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439711(CHEMBL2418954)
Affinity DataIC50:  100nMAssay Description:Inhibition of PI3Kdelta (unknown origin) using 1alpha-phosphotidylinositol by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439729(CHEMBL2418961)
Affinity DataIC50:  110nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439720(CHEMBL2418955)
Affinity DataIC50:  110nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439724(CHEMBL2418950)
Affinity DataIC50:  260nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439711(CHEMBL2418954)
Affinity DataIC50:  270nMAssay Description:Inhibition of PI3Kbeta (unknown origin) using 1alpha-phosphotidylinositol by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439719(CHEMBL2418956)
Affinity DataIC50:  790nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439725(CHEMBL2418949)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439718(CHEMBL2418957)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439711(CHEMBL2418954)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of VPS34 (unknown origin) using 1alpha-phosphotidylinositol by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439715(CHEMBL2418945)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439712(CHEMBL2418960)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439717(CHEMBL2418958)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439716(CHEMBL2418959)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using [gamma33P]ATP as substrate by top counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439712(CHEMBL2418960)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) using 1alpha-phosphotidylinositol by luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439712(CHEMBL2418960)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of PI3Kbeta (unknown origin) using 1alpha-phosphotidylinositol by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439711(CHEMBL2418954)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439711(CHEMBL2418954)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439711(CHEMBL2418954)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439711(CHEMBL2418954)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439712(CHEMBL2418960)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of PI3Kdelta (unknown origin) using 1alpha-phosphotidylinositol by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50439712(CHEMBL2418960)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of VPS34 (unknown origin) using 1alpha-phosphotidylinositol by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed