Compile Data Set for Download or QSAR
maximum 50k data
Found 29 Enz. Inhib. hit(s) with all data for entry = 4251
TargetG1/S-specific cyclin-D1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59097(Aminopyrimidine, 10)
Affinity DataIC50:  7nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59088(PD0183812)
Affinity DataIC50:  8nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM6619(3-[(9bR)-5-oxo-1H,2H,3H,5H,9bH-benzo[a]pyrrolizin-...)
Affinity DataIC50:  96nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
TargetG1/S-specific cyclin-D1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59092(Aminopyrimidine, 2)
Affinity DataIC50:  110nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-D1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59095(Aminopyrimidine, 7)
Affinity DataIC50:  160nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59088(PD0183812)
Affinity DataIC50:  165nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59090(Pyrazol-3-yl urea)
Affinity DataIC50:  200nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59089(NSC625987)
Affinity DataIC50:  200nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59097(Aminopyrimidine, 10)
Affinity DataIC50:  220nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM50319624(Aminopyrimidine, 4 | CHEMBL1084454 | N1-(4-(2,4-Di...)
Affinity DataIC50:  230nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-D1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59091(Aminopyrimidine, 1)
Affinity DataIC50:  230nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59092(Aminopyrimidine, 2)
Affinity DataIC50:  330nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59087(CHEMBL258765 | Fasca-plysi | Fascaplysin)
Affinity DataIC50:  350nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59091(Aminopyrimidine, 1)
Affinity DataIC50:  410nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59093(Aminopyrimidine, 3)
Affinity DataIC50:  430nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-D1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59096(Aminopyrimidine, 8)
Affinity DataIC50:  430nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-D1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59094(Aminopyrimidine, 6)
Affinity DataIC50:  640nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-D1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59093(Aminopyrimidine, 3)
Affinity DataIC50:  890nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM50277583(2-amino-4-methyl-1,3-thiazol-5-yl)-N-[4-(morpholin...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59095(Aminopyrimidine, 7)
Affinity DataIC50:  1.02E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59094(Aminopyrimidine, 6)
Affinity DataIC50:  1.10E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM50319619(4-(2,4-Dimethylthiazol-5-yl)-N-(4-morpholinophenyl...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59096(Aminopyrimidine, 8)
Affinity DataIC50:  2.20E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-D1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM50277583(2-amino-4-methyl-1,3-thiazol-5-yl)-N-[4-(morpholin...)
Affinity DataIC50:  2.40E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-D1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM50319624(Aminopyrimidine, 4 | CHEMBL1084454 | N1-(4-(2,4-Di...)
Affinity DataIC50:  3.80E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-D1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM50319619(4-(2,4-Dimethylthiazol-5-yl)-N-(4-morpholinophenyl...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59090(Pyrazol-3-yl urea)
Affinity DataIC50:  2.50E+4nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59087(CHEMBL258765 | Fasca-plysi | Fascaplysin)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM59089(NSC625987)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed