Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with all data for entry = 50045319
TargetNucleotide-binding oligomerization domain-containing protein 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056694(CHEMBL3326943)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human NOD2 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056693(CHEMBL3326942)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human NOD2 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056692(CHEMBL3326941)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human NOD2 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056691(CHEMBL3326924)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human NOD2 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056690(CHEMBL3326923)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human NOD2 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056689(CHEMBL3326922)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human NOD1 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056694(CHEMBL3326943)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human NOD1 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056693(CHEMBL3326942)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human NOD1 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056692(CHEMBL3326941)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human NOD1 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056691(CHEMBL3326924)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human NOD1 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056690(CHEMBL3326923)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human NOD1 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056689(CHEMBL3326922)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human NOD2 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056705(CHEMBL3326944)
Affinity DataEC50:  5.01E+3nMAssay Description:Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056704(CHEMBL3326940)
Affinity DataEC50:  7.12E+3nMAssay Description:Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056703(CHEMBL3326939)
Affinity DataEC50:  1.65E+3nMAssay Description:Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056702(CHEMBL3326934)
Affinity DataEC50:  3.74E+3nMAssay Description:Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056701(CHEMBL3326933)
Affinity DataEC50:  6.61E+3nMAssay Description:Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056700(CHEMBL3326932)
Affinity DataEC50:  7.21E+3nMAssay Description:Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056699(CHEMBL3326931)
Affinity DataEC50:  4.57E+3nMAssay Description:Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056698(CHEMBL3326930)
Affinity DataEC50:  1.13E+3nMAssay Description:Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056697(CHEMBL3326925)
Affinity DataEC50:  3.16E+3nMAssay Description:Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056696(CHEMBL2270741)
Affinity DataEC50:  3.96E+3nMAssay Description:Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056695(CHEMBL3326918)
Affinity DataEC50:  3.23E+3nMAssay Description:Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50056706(CHEMBL3326946)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM62988((1-butylbenzimidazol-2-yl)amine;hydrochloride | 1-...)
Affinity DataEC50:  7.30E+3nMAssay Description:Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed