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Found 13 Enz. Inhib. hit(s) with all data for entry = 50045436
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  24nMAssay Description:Inhibition of wild type HIV1 p66/p51 reverse transcriptase by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50062568(CHEMBL3397653)
Affinity DataIC50:  46nMAssay Description:Inhibition of wild type HIV1 p66/p51 reverse transcriptase by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50062607(CHEMBL3397650)
Affinity DataIC50:  83nMAssay Description:Inhibition of wild type HIV1 p66/p51 reverse transcriptase by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50062602(CHEMBL3397637)
Affinity DataIC50:  120nMAssay Description:Inhibition of wild type HIV1 p66/p51 reverse transcriptase by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50062567(CHEMBL3397652)
Affinity DataIC50:  160nMAssay Description:Inhibition of wild type HIV1 p66/p51 reverse transcriptase by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50062605(CHEMBL3397645)
Affinity DataIC50:  540nMAssay Description:Inhibition of wild type HIV1 p66/p51 reverse transcriptase by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of wild type HIV1 p66/p51 reverse transcriptase by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50062571(CHEMBL3397657)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of wild type HIV1 p66/p51 reverse transcriptase by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50062569(CHEMBL3397656)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of wild type HIV1 p66/p51 reverse transcriptase by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50062606(CHEMBL3397649)
Affinity DataIC50:  1.89E+4nMAssay Description:Inhibition of wild type HIV1 p66/p51 reverse transcriptase by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50062603(CHEMBL3397639)
Affinity DataIC50:  2.39E+4nMAssay Description:Inhibition of wild type HIV1 p66/p51 reverse transcriptase by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50062604(CHEMBL3397641)
Affinity DataIC50:  2.46E+4nMAssay Description:Inhibition of wild type HIV1 p66/p51 reverse transcriptase by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50062601(CHEMBL3397636)
Affinity DataIC50:  2.69E+4nMAssay Description:Inhibition of wild type HIV1 p66/p51 reverse transcriptase by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed