Compile Data Set for Download or QSAR
maximum 50k data
Found 84 Enz. Inhib. hit(s) with all data for entry = 50046011
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090950(CHEMBL3582008)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090950(CHEMBL3582008)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090950(CHEMBL3582008)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50234418((2,3-Dichloro-phenyl)-[5-methoxy-2-methyl-3-(2-mor...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090922(CHEMBL3582012)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090956(CHEMBL3582027)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090955(CHEMBL3582026)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090953(CHEMBL3582024)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090922(CHEMBL3582012)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090953(CHEMBL3582024)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090949(CHEMBL3582009)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090954(CHEMBL3582025)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090949(CHEMBL3582009)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090963(CHEMBL3582018 | US9290451, 86)
Affinity DataKi:  179nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090963(CHEMBL3582018 | US9290451, 86)
Affinity DataKi:  245nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090956(CHEMBL3582027)
Affinity DataKi:  264nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090955(CHEMBL3582026)
Affinity DataKi:  294nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090954(CHEMBL3582025)
Affinity DataKi:  352nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090957(CHEMBL3582028)
Affinity DataKi:  403nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090964(CHEMBL3582019)
Affinity DataKi:  403nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090957(CHEMBL3582028)
Affinity DataKi:  416nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090946(CHEMBL3582010)
Affinity DataKi:  421nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090960(CHEMBL3582015)
Affinity DataKi:  466nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090960(CHEMBL3582015)
Affinity DataKi:  504nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090964(CHEMBL3582019)
Affinity DataKi:  774nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090946(CHEMBL3582010)
Affinity DataKi:  902nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090923(CHEMBL3582013)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090959(CHEMBL3582021)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090958(CHEMBL3582011)
Affinity DataKi:  2.07E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090961(CHEMBL3582016)
Affinity DataKi:  2.23E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090938(CHEMBL3582014)
Affinity DataKi:  2.28E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090961(CHEMBL3582016)
Affinity DataKi:  2.87E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090959(CHEMBL3582021)
Affinity DataKi:  3.03E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090923(CHEMBL3582013)
Affinity DataKi:  3.11E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090951(CHEMBL3582022)
Affinity DataKi:  3.96E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090958(CHEMBL3582011)
Affinity DataKi:  5.26E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090965(CHEMBL3582020)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090965(CHEMBL3582020)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090952(CHEMBL3582023)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090951(CHEMBL3582022)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090938(CHEMBL3582014)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090952(CHEMBL3582023)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090950(CHEMBL3582008)
Affinity DataEC50:  4.40nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090957(CHEMBL3582028)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at human CB1 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090946(CHEMBL3582010)
Affinity DataEC50:  281nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090958(CHEMBL3582011)
Affinity DataEC50:  444nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090922(CHEMBL3582012)
Affinity DataEC50:  4.40nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090923(CHEMBL3582013)
Affinity DataEC50:  67nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090938(CHEMBL3582014)
Affinity DataEC50:  155nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50090960(CHEMBL3582015)
Affinity DataEC50:  1.81E+3nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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