Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 179nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 245nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 264nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 294nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 352nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 403nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 403nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 416nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 421nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 466nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 504nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 774nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 902nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.02E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.05E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.07E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.23E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.28E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.87E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 3.03E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.11E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 3.96E+3nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.26E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 4.40nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at human CB1 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 281nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 444nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 4.40nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 67nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 155nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 1.81E+3nMAssay Description:Activity at human CB2 receptor expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins by time-resolved FRET assayMore data for this Ligand-Target Pair