Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50046409
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM159695(US9035059, 14-18)
Affinity DataIC50:  147nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM159694(US9035059, 14-16)
Affinity DataIC50:  164nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM159693(US9035059, 14-9)
Affinity DataIC50:  168nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110678(CHEMBL3605830)
Affinity DataIC50:  547nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110581(CHEMBL3605819)
Affinity DataIC50:  594nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110697(CHEMBL3605820)
Affinity DataIC50:  685nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110688(CHEMBL3605824)
Affinity DataIC50:  733nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110691(CHEMBL3605821)
Affinity DataIC50:  1.11E+3nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Mus musculus)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110518(CHEMBL3605835)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of mouse recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Mus musculus)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110581(CHEMBL3605819)
Affinity DataIC50:  1.31E+3nMAssay Description:Inhibition of mouse recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110518(CHEMBL3605835)
Affinity DataIC50:  1.52E+3nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110679(CHEMBL3605829)
Affinity DataIC50:  1.98E+3nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110589(CHEMBL3605833)
Affinity DataIC50:  2.12E+3nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110684(CHEMBL3605825)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110689(CHEMBL3605822)
Affinity DataIC50:  2.49E+3nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110588(CHEMBL3605834)
Affinity DataIC50:  3.06E+3nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110683(CHEMBL3605826)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110680(CHEMBL3605828)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50110637(CHEMBL3605832)
Affinity DataIC50:  8.07E+3nMAssay Description:Inhibition of human recombinant MGAT2 assessed as reduction in enzyme-mediated deacylation of oleoyl-CoA incubated for 20 mins by CPM dye based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed