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Found 6 Enz. Inhib. hit(s) with all data for entry = 50046801
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50131815(CHEMBL3634608)
Affinity DataIC50:  10nMAssay Description:Inhibition of human Nav1.7 by patch-clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50132410(CHEMBL3634604)
Affinity DataIC50:  60nMAssay Description:inhibitory concentration needed to to reduce the bovine GGTase-catalyzed incorporation of [3H]-FPP into a biotin-linked K-ras (B) decapeptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50131818(CHEMBL3634605)
Affinity DataIC50:  90nMAssay Description:Inhibition of [3H]-FPP incorporation into biotin-linked K-ras decapeptide (CVIM) by bovine farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50132471(CHEMBL3634603)
Affinity DataIC50:  150nMAssay Description:inhibitory concentration needed to to reduce the bovine GGTase-catalyzed incorporation of [3H]-FPP into a biotin-linked K-ras (B) decapeptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50131817(CHEMBL3634606)
Affinity DataIC50:  400nMAssay Description:Inhibition of human Nav1.7 by patch-clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50131816(CHEMBL3634607)
Affinity DataIC50:  2.36E+3nMAssay Description:Inhibition of human Nav1.7 by patch-clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed