TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Gause Institute Of New Antibiotics
Curated by ChEMBL
Gause Institute Of New Antibiotics
Curated by ChEMBL
Affinity DataIC50: 3.93E+3nMAssay Description:Inhibition of human recombinant SIRT1 deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC as substrate incubated for 45 mins by fluorescen...More data for this Ligand-Target Pair