Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50047369
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163296(CHEMBL3793911)
Affinity DataKi:  990nMAssay Description:Binding affinity to human IP receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163296(CHEMBL3793911)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human EP4 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163296(CHEMBL3793911)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human EP2 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163296(CHEMBL3793911)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human EP1 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163296(CHEMBL3793911)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human EP3 receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163296(CHEMBL3793911)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human TP receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163296(CHEMBL3793911)
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human FP receptor by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163291(CHEMBL3793903)
Affinity DataIC50:  13nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163296(CHEMBL3793911)
Affinity DataIC50:  130nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163292(CHEMBL3794451)
Affinity DataIC50:  320nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163306(CHEMBL3793117)
Affinity DataIC50:  430nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163293(CHEMBL3793265)
Affinity DataIC50:  440nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163051(CHEMBL3793336)
Affinity DataIC50:  740nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163297(CHEMBL3793345)
Affinity DataIC50:  900nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163298(CHEMBL3793291)
Affinity DataIC50: >1.00E+3nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163305(CHEMBL3792615)
Affinity DataIC50:  1.00E+3nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163304(CHEMBL3792456)
Affinity DataIC50: >1.00E+3nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163303(CHEMBL3793247)
Affinity DataIC50: >1.00E+3nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163302(CHEMBL3794058)
Affinity DataIC50: >1.00E+3nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163301(CHEMBL3794570)
Affinity DataIC50: >1.00E+3nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163299(CHEMBL3794283)
Affinity DataIC50: >1.00E+3nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163300(CHEMBL3793957)
Affinity DataIC50: >1.00E+3nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163295(CHEMBL3793824)
Affinity DataIC50:  3.20E+3nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163150(CHEMBL3794245)
Affinity DataIC50:  2.00E+4nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163294(CHEMBL3793541)
Affinity DataIC50:  2.30E+4nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163148(CHEMBL3793417)
Affinity DataIC50: >3.00E+4nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50163215(CHEMBL3792777)
Affinity DataIC50: >3.00E+4nMAssay Description:Agonist activity at human IP receptor in platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation preincubated for 1 min follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed