Affinity DataIC50: 0.398nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by turbidimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.794nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by turbidimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]-2-Mes-ADP from human P2Y12 receptor by beta-counter analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by turbidimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Displacement of [3H]-2-Mes-ADP from human P2Y12 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of ADP-induced platelet aggregation measured for 5 mins by lig...More data for this Ligand-Target Pair
Affinity DataIC50: <10nMAssay Description:Displacement of [3H]-2-Mes-ADP from human P2Y12 receptor in platelets by scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Displacement of [3H]-2-Mes-ADP from human P2Y12 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Binding affinity to P2Y12 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Binding affinity to P2Y12 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at P2Y12 receptor (unknown origin) by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Antagonist activity at P2Y12 receptor in human washed platelets assessed as inhibition of ADP-induced platelet aggregation measured for 5 mins by lig...More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Binding affinity to P2Y12 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+5nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by turbidimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.16E+5nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by turbidimetric methodMore data for this Ligand-Target Pair