Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50048769
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50101816(CHEBI:8107 | Dilabid | Dilantin | Dilantin-125 | D...)
Affinity DataIC50:  4.00E+4nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50003659(5H-dibenzo[b,f]azepine-5-carboxamide | CARBAMAZEPI...)
Affinity DataIC50:  1.31E+5nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50227234(CHEMBL1169568)
Affinity DataIC50:  1.60E+5nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50227240(CHEMBL70727)
Affinity DataIC50:  3.80E+5nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50227231(CHEMBL41666)
Affinity DataIC50:  5.00E+5nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50227237(CHEMBL305109)
Affinity DataIC50:  5.90E+5nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50227230(CHEMBL72482)
Affinity DataIC50:  6.40E+5nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50227238(CHEMBL40727)
Affinity DataIC50: >8.00E+5nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50227235(CHEMBL68312)
Affinity DataIC50: >8.00E+5nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50227233(CHEMBL72245)
Affinity DataIC50: >8.00E+5nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50227232(CHEMBL62321)
Affinity DataIC50: >8.00E+5nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50227236(CHEMBL443266)
Affinity DataIC50: >8.00E+5nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50227229(CHEMBL62653)
Affinity DataIC50: >8.00E+5nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama

Curated by ChEMBL
LigandPNGBDBM50227239(Tridione | Trimethadione | Troxidone)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibition of [3H]-BTX-B binding to sodium channels in rat brain synapto-neurosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed