TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Inhibition of human BRAF V600E mutant using MEK1 (K97R) as substrate after 40 mins in presence of [gamma33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair