Compile Data Set for Download or QSAR
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Found 87 Enz. Inhib. hit(s) with all data for entry = 50012689
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559431(CHEMBL4753310)
Affinity DataIC50:  8nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559434(CHEMBL4784095)
Affinity DataIC50:  12nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559423(CHEMBL4744992)
Affinity DataIC50:  24nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559422(CHEMBL4778645)
Affinity DataIC50:  33nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559430(CHEMBL4753641)
Affinity DataIC50:  35nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559435(CHEMBL4754584)
Affinity DataIC50:  39nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559429(CHEMBL4758113)
Affinity DataIC50:  45nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559441(CHEMBL4783382)
Affinity DataIC50:  50nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559432(CHEMBL4762965)
Affinity DataIC50:  50nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559421(CHEMBL4754908)
Affinity DataIC50:  53nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559419(CHEMBL4749547)
Affinity DataIC50:  53nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559420(CHEMBL4784092)
Affinity DataIC50:  67nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559425(CHEMBL4755895)
Affinity DataIC50:  71nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559439(CHEMBL4793809)
Affinity DataIC50:  80nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559436(CHEMBL4799926)
Affinity DataIC50:  83nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559433(CHEMBL4759538)
Affinity DataIC50:  84nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559424(CHEMBL4798047)
Affinity DataIC50:  85nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559437(CHEMBL4745961)
Affinity DataIC50:  85nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559440(CHEMBL4757583)
Affinity DataIC50:  118nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559438(CHEMBL4758690)
Affinity DataIC50:  132nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559428(CHEMBL4754031)
Affinity DataIC50:  142nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559420(CHEMBL4784092)
Affinity DataIC50:  150nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559427(CHEMBL4788258)
Affinity DataIC50:  186nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559418(CHEMBL4777114)
Affinity DataIC50:  200nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559426(CHEMBL4753218)
Affinity DataIC50:  222nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559434(CHEMBL4784095)
Affinity DataIC50:  720nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559442(CHEMBL4744126)
Affinity DataIC50:  800nMAssay Description:Inhibition of JNK3alpha1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559423(CHEMBL4744992)
Affinity DataIC50:  810nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559432(CHEMBL4762965)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559430(CHEMBL4753641)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559431(CHEMBL4753310)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559423(CHEMBL4744992)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559435(CHEMBL4754584)
Affinity DataIC50:  1.51E+3nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559432(CHEMBL4762965)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559422(CHEMBL4778645)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559431(CHEMBL4753310)
Affinity DataIC50:  2.02E+3nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559435(CHEMBL4754584)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559425(CHEMBL4755895)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559419(CHEMBL4749547)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559433(CHEMBL4759538)
Affinity DataIC50:  2.77E+3nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559439(CHEMBL4793809)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559429(CHEMBL4758113)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559441(CHEMBL4783382)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559433(CHEMBL4759538)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559422(CHEMBL4778645)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559436(CHEMBL4799926)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559437(CHEMBL4745961)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559428(CHEMBL4754031)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559430(CHEMBL4753641)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Reaction Biology

Curated by ChEMBL
LigandPNGBDBM50559438(CHEMBL4758690)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate after 22 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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