Compile Data Set for Download or QSAR
maximum 50k data
Found 40 Enz. Inhib. hit(s) with all data for entry = 50013208
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50:  4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50235334(CHEMBL4070391)
Affinity DataIC50:  22nMAssay Description:Inhibition of CDK2/cyclin A2 (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50235334(CHEMBL4070391)
Affinity DataIC50:  31nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563675(CHEMBL4762791)
Affinity DataIC50:  660nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563675(CHEMBL4762791)
Affinity DataIC50:  680nMAssay Description:Inhibition of CDK2/cyclin A2 (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563673(CHEMBL4797166)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563688(CHEMBL4761406)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563669(CHEMBL4755169)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563690(CHEMBL4745418)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563674(CHEMBL4794743)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563675(CHEMBL4762791)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of CDK1/cyclin B (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50235334(CHEMBL4070391)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of CDK1/cyclin B (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563683(CHEMBL4749217)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563687(CHEMBL4788506)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563668(CHEMBL4783322)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563672(CHEMBL4744723)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563681(CHEMBL4759594)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563694(CHEMBL4740445)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATP b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563689(CHEMBL4796499)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563667(CHEMBL4742100)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50235334(CHEMBL4070391)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563675(CHEMBL4762791)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563682(CHEMBL4785267)
Affinity DataIC50: >1.25E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563670(CHEMBL4742111)
Affinity DataIC50: >1.25E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563678(CHEMBL4781962)
Affinity DataIC50:  1.42E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563675(CHEMBL4762791)
Affinity DataIC50:  1.43E+4nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563671(CHEMBL4788230)
Affinity DataIC50:  1.78E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50235334(CHEMBL4070391)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563680(CHEMBL4754214)
Affinity DataIC50:  2.44E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563686(CHEMBL4753339)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563679(CHEMBL4761946)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563676(CHEMBL4750349)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563684(CHEMBL4789416)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563692(CHEMBL4785238)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563691(CHEMBL4764317)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563685(CHEMBL4745984)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563677(CHEMBL4743433)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563693(CHEMBL4795420)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) using peptide substrate in presence of [gamma33P]ATP by image analyserMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataKd:  18nMAssay Description:Binding affinity to CDK2 (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Institute For Organic Syntheses (Vuos)

Curated by ChEMBL
LigandPNGBDBM50563675(CHEMBL4762791)
Affinity DataKd:  4.10E+3nMAssay Description:Binding affinity to CDK2 (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB