Affinity DataKi: 3.30nMAssay Description:Displacement of 3 nM [3H]Nalpha-methylhistamine from human H3R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Displacement of 40 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of 10 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Displacement of 10 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Displacement of 2 nM [3H]UR-PI294 from human H3R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Displacement of 2 nM [3H]UR-PI294 from human H3R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of 10 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of 40 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to human H4RMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of 3 nM [3H]Nalpha-methylhistamine from human H3R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of 2 nM [3H]UR-PI294 from human H3R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of 3 nM [3H]Nalpha-methylhistamine from human H3R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of 40 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of 10 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Displacement of 40 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Displacement of 10 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:Displacement of 10 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 145nMAssay Description:Displacement of 3 nM [3H]Nalpha-methylhistamine from human H3R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 186nMAssay Description:Displacement of 10 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 204nMAssay Description:Displacement of 10 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 204nMAssay Description:Displacement of 3 nM [3H]Nalpha-methylhistamine from human H3R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 204nMAssay Description:Displacement of 2 nM [3H]UR-PI294 from human H3R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 204nMAssay Description:Displacement of 40 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 309nMAssay Description:Displacement of 40 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 355nMAssay Description:Displacement of [3H]-UR-DEBa176 from human H4R expressed in HEK293T-SF-His6-CRE-Luc cellsMore data for this Ligand-Target Pair
Affinity DataKi: 447nMAssay Description:Displacement of 40 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Displacement of [3H]-UR-DEBa176 from mouse H4R expressed in HEK293T-SF-His6-CRE-Luc cellsMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Displacement of [3H]UR-PI294 from human H3R expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Displacement of [3H]UR-PI294 from human H3R expressed in human SK-N-MC-cellsMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Displacement of [3H]UR-PI294 from human H3R expressed in Sf9 cells co-expressing Galphai2 and Gbeta1gamma2More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Displacement of [3H]histamine from human H3R expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Displacement of [3H]UR-PI294 from human H3R expressed in Sf9 cells co-expressing RGS19 and Galphai2 and Gbeta1gamma2More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Displacement of [3H]histamine from human H3R expressed in Sf9 cells co-expressing RGS19 and Galpha1 and Gbeta1gamma2More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Displacement of [3H]histamine from human H3R expressed in Sf9 cells co-expressing Galpha1 and Gbeta1gamma2More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Displacement of [3H]histamine from human H3R expressed in human SK-N-MC-cellsMore data for this Ligand-Target Pair
Affinity DataKi: 537nMAssay Description:Displacement of 2 nM [3H]UR-PI294 from human H3R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 562nMAssay Description:Displacement of 20 nM [3H]UR-DE257 from human H2R expressed in Sf9 cell membranes co-expressing GsalphaS by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 617nMAssay Description:Displacement of 10 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 692nMAssay Description:Displacement of 3 nM [3H]Nalpha-methylhistamine from human H3R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition bind...More data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of 20 nM [3H]UR-DE257 from human H2R expressed in Sf9 cell membranes co-expressing GsalphaS by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of 20 nM [3H]UR-DE257 from human H2R expressed in Sf9 cell membranes co-expressing GsalphaS by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of 5 nM [3H-pyrilamine from human H1R expressed in Sf9 cell membranes co-expressing RGS4 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of 20 nM [3H]UR-DE257 from human H2R expressed in Sf9 cell membranes co-expressing GsalphaS by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of 5 nM [3H-pyrilamine from human H1R expressed in Sf9 cell membranes co-expressing RGS4 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of 5 nM [3H-pyrilamine from human H1R expressed in Sf9 cell membranes co-expressing RGS4 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of 20 nM [3H]UR-DE257 from human H2R expressed in Sf9 cell membranes co-expressing GsalphaS by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of 20 nM [3H]UR-DE257 from human H2R expressed in Sf9 cell membranes co-expressing GsalphaS by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.12E+3nMAssay Description:Displacement of 3 nM [3H]Nalpha-methylhistamine from human H3R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 1.91E+3nMAssay Description:Displacement of 40 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Displacement of [3H]-UR-DEBa176 from rat H4R expressed in HEK293T-SF-His6-CRE-Luc cellsMore data for this Ligand-Target Pair