Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 50032992
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337589(3-(3-(4-(6-phenylhexyloxy)phenyl)propylamino)propa...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337599((E/Z)-3-(3-(4-(3-phenylpropoxy)phenyl)allylamino)p...)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337591(3-(3-(4-(3-phenylpropoxy)phenyl)propylamino)propan...)
Affinity DataEC50:  9.00E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337592(3-(3-(4-(5-phenylpentyloxy)phenyl)propylamino)prop...)
Affinity DataEC50:  4.20E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 2(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337592(3-(3-(4-(5-phenylpentyloxy)phenyl)propylamino)prop...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P2 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337593(CHEMBL1683051 | trans-3-(3-(4-(3-phenylpropoxy)ben...)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337594(3-(4-(4-(3-phenylpropoxy)phenyl)piperidin-1-yl)pro...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337595(3-(4-(4-(3-phenylpropoxy)phenyl)-5,6-dihydropyridi...)
Affinity DataEC50:  45nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337596(CHEMBL1683048 | cis-3-(3-(4-(3-phenylpropoxy)pheny...)
Affinity DataEC50:  930nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337597(CHEMBL1683047 | trans-3-(3-(4-(3-phenylpropoxy)phe...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337598(CHEMBL1683046 | trans-3-(2-methyl-3-(4-(3-phenylpr...)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337599((E/Z)-3-(3-(4-(3-phenylpropoxy)phenyl)allylamino)p...)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337589(3-(3-(4-(6-phenylhexyloxy)phenyl)propylamino)propa...)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337590(3-(3-(4-(4-phenylbutoxy)phenyl)propylamino)propano...)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337591(3-(3-(4-(3-phenylpropoxy)phenyl)propylamino)propan...)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337592(3-(3-(4-(5-phenylpentyloxy)phenyl)propylamino)prop...)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337592(3-(3-(4-(5-phenylpentyloxy)phenyl)propylamino)prop...)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human S1P5 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337593(CHEMBL1683051 | trans-3-(3-(4-(3-phenylpropoxy)ben...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337594(3-(4-(4-(3-phenylpropoxy)phenyl)piperidin-1-yl)pro...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337595(3-(4-(4-(3-phenylpropoxy)phenyl)-5,6-dihydropyridi...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337596(CHEMBL1683048 | cis-3-(3-(4-(3-phenylpropoxy)pheny...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337597(CHEMBL1683047 | trans-3-(3-(4-(3-phenylpropoxy)phe...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337598(CHEMBL1683046 | trans-3-(2-methyl-3-(4-(3-phenylpr...)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50337590(3-(3-(4-(4-phenylbutoxy)phenyl)propylamino)propano...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO cells assessed as intracellular calcium levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed