Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50005381
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50036267(CHEMBL268874 | Dyn A(H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg...)
Affinity DataIC50:  0.580nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 1 in guinea pig brain using [3H]-U-69,593 as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50138774(CHEMBL415795 | Linear [D-Ala3]Dyn A-(1-11)NH2)
Affinity DataIC50:  0.760nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 1 in guinea pig brain using [3H]-U-69,593 as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50036266(CHEMBL262963 | Dyn A(H-Tyr-Gly-Ala-Phe-Leu-Arg-Arg...)
Affinity DataIC50:  1.10nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 1 in guinea pig brain using [3H]-U-69,593 as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50036267(CHEMBL268874 | Dyn A(H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg...)
Affinity DataIC50:  9.90nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 in guinea pig brain using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50036267(CHEMBL268874 | Dyn A(H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg...)
Affinity DataIC50:  26nMAssay Description:Compound was evaluated for its receptor binding affinity at[3H]cyclo[D-pen2,p-cl-Phe4,D-Pen5](delta receptor) to opoid receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50036266(CHEMBL262963 | Dyn A(H-Tyr-Gly-Ala-Phe-Leu-Arg-Arg...)
Affinity DataIC50:  210nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 in guinea pig brain using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50138774(CHEMBL415795 | Linear [D-Ala3]Dyn A-(1-11)NH2)
Affinity DataIC50:  260nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 in guinea pig brain using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50036266(CHEMBL262963 | Dyn A(H-Tyr-Gly-Ala-Phe-Leu-Arg-Arg...)
Affinity DataIC50:  730nMAssay Description:Compound was evaluated for its receptor binding affinity at[3H]cyclo[D-pen2,p-cl-Phe4,D-Pen5](delta receptor) to opoid receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50138774(CHEMBL415795 | Linear [D-Ala3]Dyn A-(1-11)NH2)
Affinity DataIC50:  1.00E+3nMAssay Description:Compound was evaluated for its receptor binding affinity at[3H]cyclo[D-pen2,p-cl-Phe4,D-Pen5](delta receptor) to opoid receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed