Compile Data Set for Download or QSAR
maximum 50k data
Found 136 Enz. Inhib. hit(s) with all data for entry = 4978
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82255(D-Phe-Cys-Tyr-D-Trp-Lys-Abu-Cys-Nal-NH | NC8-12)
Affinity DataKi:  0.0240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.0260nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84628(EC5-21)
Affinity DataKi:  0.0280nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82255(D-Phe-Cys-Tyr-D-Trp-Lys-Abu-Cys-Nal-NH | NC8-12)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50097783(CHEMBL438401 | D-Trp8 SST-14 | SOMATOSTATIN | SRIF...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50097783(CHEMBL438401 | D-Trp8 SST-14 | SOMATOSTATIN | SRIF...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84621(BIM 23042)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82462(BIM 23059 | D-Nal-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Thr...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84620(DC23-60)
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50097783(CHEMBL438401 | D-Trp8 SST-14 | SOMATOSTATIN | SRIF...)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82462(BIM 23059 | D-Nal-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Thr...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84618(Leu8, D-Trp22, Tyr25 SST-28)
Affinity DataKi:  0.410nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82465(BIM 23023 | BIM-23023 | D-Phe-L-Cys(1)-L-Tyr-D-Trp...)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82465(BIM 23023 | BIM-23023 | D-Phe-L-Cys(1)-L-Tyr-D-Trp...)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.530nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  0.620nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50097783(CHEMBL438401 | D-Trp8 SST-14 | SOMATOSTATIN | SRIF...)
Affinity DataKi:  0.630nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82459(BIM 23058 | BIM-23058 | D-Phe-L-Phe-L-Tyr-D-Trp-L-...)
Affinity DataKi:  0.670nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84624(BIM 23068)
Affinity DataKi:  0.710nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84630(BIM 23060)
Affinity DataKi:  0.710nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84628(EC5-21)
Affinity DataKi:  0.970nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84621(BIM 23042)
Affinity DataKi:  1.15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82459(BIM 23058 | BIM-23058 | D-Phe-L-Phe-L-Tyr-D-Trp-L-...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50063819(BIM 23050 | CHEMBL413535 | cyclo[NMeDAla-Tyr-DTrp-...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81766(CAS_3086456 | MK 678 | NSC_3086456)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84624(BIM 23068)
Affinity DataKi:  1.54nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84624(BIM 23068)
Affinity DataKi:  1.55nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM81766(CAS_3086456 | MK 678 | NSC_3086456)
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  2.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84623(NC4-28B)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84630(BIM 23060)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84626(BIM 23034)
Affinity DataKi:  2.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84620(DC23-60)
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84626(BIM 23034)
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  4.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84623(NC4-28B)
Affinity DataKi:  4.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  4.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Mcgill University

Curated by PDSP Ki Database
LigandPNGBDBM84622(BIM 23057)
Affinity DataKi:  4.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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